SCHEMBL18092002

SCHEMBL18092002

CCCCc1noc(C)c1/C=C\c1nc(C)c(OC(=O)NCCO)s1

nearest known ligand 0.32

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.32
ALOX5 P09917 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18091990 1.00 ALDH1A1 (0.32) ALDH1A1ALOX5
SCHEMBL18092007 0.88 TP53 (0.31) ALOX5
SCHEMBL18092069 0.87
SCHEMBL18092001 0.87 TP53 (0.30)
SCHEMBL18091976 0.86 ACACB (0.34)
SCHEMBL18091988 0.86
SCHEMBL18092064 0.86 GABRA5 (0.30)
SCHEMBL18092052 0.85
SCHEMBL18092078 0.85
SCHEMBL18092071 0.84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427459-B1 ISOXAZOLE-THIAZOLE DERIVATIVES AS GABA A RECEPTOR INVERSE AGONISTS FOR USE IN THE TREATMENT OF COGNITIVE DISORDERS HOFFMANN LA ROCHE (CH) 2016-09-28 EP claimed