SCHEMBL18106903

SCHEMBL18106903

O=C(O)Nc1nc2ccccc2[nH]1.O=[N+]([O-])c1cccc(C2CC2)c1

nearest known ligand 0.62

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 9/20 0.62
SMN1; SMN2 Q16637 8/20 0.62
NPC1 O15118 6/20 0.62
RAB9A P51151 5/20 0.62
ALDH1A1 P00352 2/20 0.62
KMT2A Q03164 3/20 0.54
MAPT P10636 3/20 0.54
MEN1 O00255 2/20 0.54
LPAR2 Q9HBW0 1/20 0.48
TDP1 Q9NUW8 2/20 0.47
POLB P06746 1/20 0.47
MCL1 Q07820 1/20 0.47
KDM4E B2RXH2 1/20 0.47
CYP1A2 P05177 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18106906 0.84 SMN1; SMN2 (0.63) SMN1; SMN2NPC1RAB9AALDH1A1KMT2A
SCHEMBL18106895 0.84 LPAR2 (0.67) SMN1; SMN2NPC1RAB9AKMT2AMAPT
SCHEMBL18106896 0.83 NPC1 (0.60) SMN1; SMN2NPC1RAB9AKMT2AMEN1
SCHEMBL18106909 0.83 RAB9A (0.60) SMN1; SMN2NPC1RAB9AALDH1A1KMT2A
SCHEMBL15944972 0.81 LPAR2 (0.71) IRAK4SMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL18106900 0.79 SMN1; SMN2 (0.48) IRAK4SMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL18106907 0.77 NPC1 (0.60) SMN1; SMN2NPC1RAB9AALDH1A1KMT2A
SCHEMBL3597174 0.77 IRAK4 (1.00) IRAK4SMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL30933802 0.76 IRAK4 (0.70) IRAK4SMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL25956566 0.76 IRAK4 (0.70) IRAK4SMN1; SMN2NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2742029-B1 N-(BENZIMIMDAZOL-2-YL)-CYCLOPROPANE CARBOXAMIDES AS LYSOPHOSPHATIDIC ACID ANTAGONISTS MERCK PATENT GMBH (DE) 2016-10-05 EP claimed