SCHEMBL1812949

SCHEMBL1812949

CCCCc1ccc(C#Cc2ccc(CNCc3ccc(OC(C)C(=O)O)cc3)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACACB O00763 10/20 0.49
ADRB3 P13945 5/20 0.47
S1PR2 O95136 1/20 0.46
S1PR4 O95977 1/20 0.46
S1PR1 P21453 1/20 0.46
S1PR3 Q99500 1/20 0.46
MMP2 P08253 1/20 0.45
MMP9 P14780 1/20 0.45
EPHX2 P34913 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1817481 0.99 ACACB (0.48) ACACBADRB3S1PR2S1PR4S1PR1
SCHEMBL4465853 0.85 FFAR1 (0.53) ACACBADRB3S1PR2S1PR4S1PR1
SCHEMBL1810232 0.82 MMP2 (0.47) ACACBMMP2MMP9
SCHEMBL2858029 0.82 FFAR1 (0.54) ACACBS1PR2S1PR4S1PR1S1PR3
SCHEMBL1814796 0.82 PTGES (0.53) ACACBADRB3MMP2MMP9EPHX2
Hydrochloric Acid SCHEMBL4469874 0.81 FFAR1 (0.52) ACACBS1PR2S1PR4S1PR1S1PR3
SCHEMBL28378269 0.80 PPARA (0.62) ADRB3S1PR2S1PR1
SCHEMBL28575461 0.80 PPARA (0.62) ADRB3S1PR2S1PR1
SCHEMBL28379854 0.80 PPARA (0.62) ADRB3S1PR2S1PR1
SCHEMBL2858924 0.79 RARB (0.61) ACACBS1PR2S1PR4S1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7947851-B2 1,1′-(1,2-ethynediyl)bis-benzene derivatives as PTP 1-B inhibitors MERCK SERONO SA (CH) 2011-05-24 US disclosed