SCHEMBL18153393

SCHEMBL18153393

Cc1cc(N2CCN(C(=O)O)CC2)nc(Cl)n1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 17/20 0.51
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
HRH4 Q9H3N8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21193554 0.88 GBA1 (0.66) GBA1
SCHEMBL18153268 0.84 HRH4 (0.41) GBA1LMNAHRH4
SCHEMBL18153279 0.81 GPR119 (0.56) GBA1ALDH1A1LMNAHRH4
SCHEMBL9884923 0.79 HRH4 (0.64) HRH4
SCHEMBL11963431 0.79 GBA1 (0.42) GBA1ALDH1A1LMNA
SCHEMBL3405363 0.79 CRHBP (0.61) GBA1ALDH1A1LMNAHRH4
SCHEMBL3410886 0.77 CRHBP (0.64) GBA1ALDH1A1LMNAHRH4
SCHEMBL31647387 0.77 MAPT (0.67) ALDH1A1LMNA
SCHEMBL21815386 0.76 GBA1 (0.51) GBA1ALDH1A1LMNA
SCHEMBL16795197 0.76 PHGDH (0.44) GBA1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240270737-A1 SMALL MOLECULAR INHIBITORS OF STING SIGNALING COMPOSITIONS AND METHODS OF USE STINGINN INC. (US) 2024-08-15 US disclosed
EP-4351578-A1 SMALL MOLECULAR INHIBITORS OF STING SIGNALING COMPOSITIONS AND METHODS OF USE Stinginn Inc (US) 2024-04-17 EP disclosed
WO-2022245986-A1 SMALL MOLECULAR INHIBITORS OF STING SIGNALING COMPOSITIONS AND METHODS OF USE STINGINN INC (US) 2022-11-24 WO disclosed
EP-3856737-A1 HETEROCYCLYL COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE DISEASE F. Hoffmann-La Roche AG (CH) 2021-08-04 EP disclosed
WO-2020064792-A1 HETEROCYCLYL COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE DISEASE F. HOFFMANN-LA ROCHE AG (CH) 2020-04-02 WO disclosed
EP-3283472-A1 HEPATITIS B VIRAL ASSEMBLY EFFECTORS Indiana University Research&Technology Corporation (US) 2018-02-21 EP disclosed
WO-2016168619-A1 HEPATITIS B VIRAL ASSEMBLY EFFECTORS INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION (US) 2016-10-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240270737-A1 SMALL MOLECULAR INHIBITORS OF STING SIGNALING COMPOSITIONS AND METHODS OF USE STING1, IRF3, MAVS GBA1 2243/4885ALDH1A1 4812/4885LMNA 2811/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.