SCHEMBL18155239

SCHEMBL18155239

Cc1ccc2c(c1)c1c(n2C#Cc2ccncc2)C(C)N(C)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 4/20 0.38
HTR6 P50406 3/20 0.38
HSD17B10 Q99714 6/20 0.34
KDM4E B2RXH2 6/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2D6 P10635 2/20 0.34
TP53 P04637 1/20 0.34
CYP3A4 P08684 1/20 0.34
HTR1A P08908 1/20 0.34
ADRA2A P08913 1/20 0.34
CHRM1 P11229 1/20 0.34
MAOA P21397 1/20 0.34
DRD1 P21728 1/20 0.34
SLC6A2 P23975 1/20 0.34
TEAD1 P28347 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18155246 0.91 HSD17B10 (0.37) HRH1HTR6HSD17B10KDM4EMEN1
SCHEMBL13654437 0.89 KDM4E (0.34) KDM4EDRD1KCNH2GAAMAPT
SCHEMBL18155267 0.88 HRH1 (0.39) HRH1HTR6HSD17B10KDM4EMEN1
SCHEMBL1120646 0.87 KDM4E (0.34) HSD17B10KDM4EMEN1KMT2ACYP1A2
SCHEMBL13663461 0.87 HTR6 (0.38) HRH1HTR6HSD17B10KDM4EMEN1
SCHEMBL18155247 0.87 HRH1 (0.38) HRH1HTR6HSD17B10KDM4EMEN1
SCHEMBL18155286 0.85 HTR6 (0.40) HRH1HTR6HSD17B10KDM4EMEN1
SCHEMBL18155259 0.85 KDM4E (0.36) HSD17B10KDM4EMEN1KMT2ACYP1A2
SCHEMBL18155277 0.83 HSD17B10 (0.33) HRH1HTR6HSD17B10KDM4EMEN1
SCHEMBL18155322 0.80 MAPT (0.32) HRH1HTR6HSD17B10KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9469641-B2 Pyrido[3,4-B]indoles and methods of use MEDIVATION TECHNOLOGIES, INC. (US) 2016-10-18 US disclosed