SCHEMBL18155286

SCHEMBL18155286

COc1ccc(C#Cn2c3c(c4cc(C)ccc42)CCN(C)C3C)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.40
HRH1 P35367 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.34
HSD17B10 Q99714 4/20 0.33
KDM4E B2RXH2 3/20 0.33
SLC6A4 P31645 2/20 0.33
DRD1 P21728 2/20 0.33
MEN1 O00255 1/20 0.33
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
KMT2A Q03164 1/20 0.33
HTR1A P08908 1/20 0.33
ADRA2A P08913 1/20 0.33
CHRM1 P11229 1/20 0.33
MAOA P21397 1/20 0.33
SLC6A2 P23975 1/20 0.33
TEAD1 P28347 1/20 0.33
SLC6A3 Q01959 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18155246 0.92 HSD17B10 (0.37) HTR6HRH1HSD17B10KDM4ESLC6A4
SCHEMBL13654699 0.90 DRD2 (0.36) HTR6L3MBTL1HSD17B10KDM4ESLC6A4
SCHEMBL13663461 0.88 HTR6 (0.38) HTR6HRH1HSD17B10KDM4ESLC6A4
SCHEMBL1120646 0.88 KDM4E (0.34) HSD17B10KDM4ESLC6A4DRD1MEN1
SCHEMBL18155270 0.87 HTR6 (0.40) HTR6HRH1L3MBTL1HSD17B10KDM4E
SCHEMBL18155322 0.86 MAPT (0.32) HTR6HRH1HSD17B10KDM4ESLC6A4
SCHEMBL18155259 0.85 KDM4E (0.36) HSD17B10KDM4ESLC6A4DRD1MEN1
SCHEMBL18155239 0.85 HRH1 (0.38) HTR6HRH1HSD17B10KDM4ESLC6A4
SCHEMBL18155277 0.84 HSD17B10 (0.33) HTR6HRH1HSD17B10KDM4ESLC6A4
SCHEMBL1120512 0.81 KDM4E (0.36) HSD17B10KDM4ESLC6A4DRD1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9469641-B2 Pyrido[3,4-B]indoles and methods of use MEDIVATION TECHNOLOGIES, INC. (US) 2016-10-18 US disclosed