SCHEMBL18156508

SCHEMBL18156508

Cc1ccc(F)c2c(=O)[nH]c(-c3ccc(C(=O)N4CCN(CCOSc5ccccc5)CC4)cc3)cc12

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 6/20 0.42
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
DRD3 P35462 2/20 0.39
DRD2 P14416 1/20 0.39
LDHA P00338 2/20 0.38
TNKS O95271 4/20 0.38
KCNH2 Q12809 1/20 0.38
ALDH1A1 P00352 2/20 0.37
PARP1 P09874 2/20 0.37
ALOX15 P16050 1/20 0.37
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16625249 0.84 ALDH1A1 (0.45) TNKSALDH1A1PARP1KDM4E
SCHEMBL16625331 0.84 KCNA5 (0.40) KCNA5MEN1KMT2ADRD3DRD2
SCHEMBL16625237 0.81 TNKS (0.52) MEN1KMT2ATNKSALDH1A1PARP1
SCHEMBL23302837 0.75 SIGMAR1 (0.47) KCNA5MEN1KMT2ADRD2KCNH2
SCHEMBL29882297 0.75 SIGMAR1 (0.47) KCNA5MEN1KMT2ADRD2KCNH2
SCHEMBL16625269 0.75 KMT2A (0.53) MEN1KMT2ATNKSPARP1
SCHEMBL16625165 0.74 TNKS (0.56) KCNA5KMT2ADRD3DRD2TNKS
SCHEMBL23302442 0.72 ACHE (0.47) DRD2LDHAKCNH2PARP1L3MBTL1
SCHEMBL16625329 0.71 TNKS (0.51) KCNA5MEN1KMT2ADRD3DRD2
SCHEMBL16625330 0.70 TNKS (0.43) KCNA5MEN1KMT2ADRD3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2822656-B1 3-ARYL-5-SUBSTITUTED-ISOQUINOLIN-1-ONE COMPOUNDS AND THEIR THERAPEUTIC USE CANCER RES INST ROYAL (GB) 2016-10-19 EP disclosed