SCHEMBL1816243

SCHEMBL1816243

c1ccc(-c2c3ccccc3c(-c3ccc(-c4cccc5c4ccc4cc6ccccc6cc45)cc3)c3ccccc23)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 9/20 0.46
ESR2 Q92731 8/20 0.46
ALDH1A1 P00352 2/20 0.42
HIF1A Q16665 1/20 0.42
CYP1B1 Q16678 1/20 0.42
HSD17B10 Q99714 1/20 0.42
SOS1 Q07889 1/20 0.42
HSD17B1 P14061 2/20 0.42
HSD17B2 P37059 2/20 0.42
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
MPI P34949 1/20 0.41
KMT2A Q03164 1/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2B6 P20813 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23242772 0.94 ESR1 (0.44) ESR1ESR2ALDH1A1HIF1ACYP1B1
SCHEMBL1817923 0.92 ESR1 (0.45) ESR1ESR2ALDH1A1HIF1ACYP1B1
SCHEMBL2455000 0.92 ESR1 (0.47) ESR1ESR2ALDH1A1HIF1ACYP1B1
SCHEMBL28606956 0.92 ESR1 (0.50) ESR1ESR2ALDH1A1HSD17B1HSD17B2
SCHEMBL2859818 0.92 ALDH1A1 (0.50) ESR1ESR2ALDH1A1HIF1ACYP1B1
SCHEMBL2991961 0.90 SOS1 (0.48) ESR1ESR2ALDH1A1SOS1HSD17B1
SCHEMBL27610205 0.90 ESR1 (0.51) ESR1ESR2ALDH1A1HIF1AHSD17B10
SCHEMBL2995209 0.90 ALDH1A1 (0.52) ALDH1A1HIF1ACYP1B1HSD17B10HSD17B1
SCHEMBL31290733 0.90 ALDH1A1 (0.52) ALDH1A1HIF1ACYP1B1HSD17B10SOS1
SCHEMBL23242753 0.90 GPR84 (0.42) ESR1ESR2ALDH1A1HIF1ACYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120217449-A1 MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2012-08-30 US disclosed
WO-2011054442-A2 MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2011-05-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120217449-A1 MATERIALS FOR ELECTRONIC DEVICES EFNA1, DDT, ERCC1 ESR1 45/4885ESR2 135/4885ALDH1A1 261/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.