SCHEMBL18166455

SCHEMBL18166455

Cc1ccc(-c2cc(OC(=O)NCc3ccncc3)cc(-n3nnnc3C(C)C)c2)c(F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 4/20 0.42
EPHX1 P07099 1/20 0.41
KDM1A O60341 2/20 0.40
HDAC1 Q13547 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.37
LMNA P02545 2/20 0.35
RECQL P46063 1/20 0.35
CDK2 P24941 1/20 0.35
GSK3B P49841 1/20 0.35
MMP2 P08253 1/20 0.34
CYP3A4 P08684 1/20 0.34
STAT3 P40763 1/20 0.34
HTT P42858 1/20 0.34
MMP13 P45452 1/20 0.34
MAPK14 Q16539 1/20 0.34
POLB P06746 1/20 0.34
ALDH1A1 P00352 1/20 0.34
FLT1 P17948 1/20 0.33
KDR P35968 1/20 0.33
PTGS2 P35354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18166296 0.91 EPHX1 (0.45) FAAHEPHX1KDM1AHDAC1SMN1; SMN2
SCHEMBL10244871 0.87 HDAC1 (0.51) KDM1AHDAC1SMN1; SMN2LMNARECQL
SCHEMBL18166367 0.87 MAOB (0.40) FAAHSMN1; SMN2
SCHEMBL18166394 0.86 ROCK1 (0.38) LMNACDK2GSK3BCYP3A4
SCHEMBL18166274 0.85 P2RX3 (0.49) FAAH
SCHEMBL18036393 0.83 P2RX3 (0.43) FAAH
SCHEMBL18036425 0.82 P2RX3 (0.35) FAAHPTGS2
SCHEMBL18036367 0.82 P2RX3 (0.35) FAAHPTGS2
SCHEMBL18166460 0.81 AKR1C3 (0.38) SMN1; SMN2CDK2GSK3BCYP3A4POLB
SCHEMBL18166380 0.80 P2RX3 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2038264-B1 TETRAZOLE-SUBSTITUTED ARYLAMIDES HOFFMANN LA ROCHE (CH) 2016-10-26 EP claimed