SCHEMBL18172020

SCHEMBL18172020

CCOC(=O)c1ccnn1-c1ccccc1OC

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.47
HSD17B10 Q99714 2/20 0.47
ALDH1A1 P00352 1/20 0.47
HPGD P15428 1/20 0.47
ALOX15 P16050 1/20 0.47
KDM4E B2RXH2 3/20 0.47
MAPT P10636 3/20 0.47
LMNA P02545 2/20 0.47
GLA P06280 1/20 0.47
HTT P42858 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
PKM P14618 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.45
NR3C2 P08235 1/20 0.44
KMT2A Q03164 2/20 0.44
TDP1 Q9NUW8 2/20 0.43
POLB P06746 1/20 0.43
APEX1 P27695 1/20 0.43
RECQL P46063 1/20 0.43
CTDSP1 Q9GZU7 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28817913 0.83 NPSR1 (0.56) ALDH1A1HPGDKDM4EMAPTNPSR1
SCHEMBL6987458 0.82 NR3C2 (0.48) ALDH1A1NPSR1L3MBTL1NR3C2KMT2A
SCHEMBL22731945 0.81 HSD11B1 (0.53) GAAHSD17B10ALDH1A1HPGDALOX15
SCHEMBL29574308 0.81 HSD11B1 (0.53) GAAHSD17B10ALDH1A1HPGDALOX15
SCHEMBL9681622 0.79 ALDH1A1 (0.57) GAAHSD17B10ALDH1A1HPGDKDM4E
SCHEMBL462999 0.78 MAPK14 (0.50) GAAHSD17B10ALDH1A1HPGDALOX15
SCHEMBL6313155 0.78 ALDH1A1 (0.53) GAAHSD17B10ALDH1A1HPGDALOX15
SCHEMBL6174962 0.78 MAPT (0.57) GAAKDM4EMAPTLMNAGLA
SCHEMBL25314471 0.76 SLC5A1 (0.42) GAAALDH1A1HPGDKDM4EMAPT
SCHEMBL17844090 0.76 ALDH1A1 (0.67) GAAHSD17B10ALDH1A1HPGDALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3286178-A1 AMINO-SUBSTITUTED HETEROCYCLIC DERIVATIVES AS SODIUM CHANNEL INHIBITORS Almirall S.A. (ES) 2018-02-28 EP disclosed
WO-2016170009-A1 AMINO-SUBSTITUTED HETEROCYCLIC DERIVATIVES AS SODIUM CHANNEL INHIBITORS ALMIRALL, S.A. (ES) 2016-10-27 WO disclosed