SCHEMBL1817267

SCHEMBL1817267

Brc1ccc(CC#Cc2ccccc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PYCR1 P32322 1/20 0.60
FFAR1 O14842 4/20 0.50
FFAR4 Q5NUL3 3/20 0.50
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
THPO P40225 1/20 0.48
BLM P54132 1/20 0.47
PMP22 Q01453 1/20 0.47
APP P05067 1/20 0.44
HTR2A P28223 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
ALDH1A1 P00352 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MAPK1 P28482 1/20 0.39
LMNA P02545 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14417894 0.92 FFAR1 (0.54) PYCR1FFAR1FFAR4CYP1A2CYP3A4
SCHEMBL13997198 0.89 PYCR1 (0.47) PYCR1FFAR1FFAR4APPHTR2A
SCHEMBL3397750 0.84 CYP1A2 (0.58) FFAR1FFAR4CYP1A2CYP3A4CYP2C9
SCHEMBL27563099 0.79 FFAR1 (0.54) FFAR1FFAR4CYP1A2CYP3A4CYP2C9
SCHEMBL8910688 0.79 POLB (0.58) PYCR1FFAR1FFAR4CYP1A2CYP3A4
SCHEMBL28772070 0.79 FFAR1 (0.50) PYCR1FFAR1FFAR4CYP1A2CYP3A4
SCHEMBL651586 0.77 APP (0.67) PYCR1FFAR1FFAR4CYP1A2CYP3A4
SCHEMBL5401236 0.77 APP (0.67) PYCR1FFAR1FFAR4CYP1A2CYP3A4
SCHEMBL28266545 0.76 PYCR1 (0.49) PYCR1FFAR1FFAR4CYP1A2CYP3A4
SCHEMBL21244052 0.75 LTA4H (0.55) FFAR1FFAR4CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2494408-A1 PHOTOCHROMIC MATERIALS Transitions Optical, Inc. (US) 2012-09-05 EP disclosed
WO-2011053615-A1 PHOTOCHROMIC MATERIALS TRANSITIONS OPTICAL, INC. (US) 2011-05-05 WO disclosed