SCHEMBL18173604

SCHEMBL18173604

CCOC(=C(C#N)C#N)c1ccc(Oc2ccccc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 2/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
HPGD P15428 1/20 0.46
CRHBP P24387 1/20 0.46
CRHR2 Q13324 1/20 0.46
PPARG P37231 1/20 0.42
PPARA Q07869 1/20 0.42
MAPK14 Q16539 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.41
PTGS2 P35354 1/20 0.40
MAPT P10636 2/20 0.40
ALDH1A1 P00352 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
PARP10 Q53GL7 1/20 0.40
HTT P42858 1/20 0.40
LMNA P02545 1/20 0.40
THRB P10828 1/20 0.40
SRD5A2 P31213 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2200157 0.87 SMN1; SMN2 (0.46) NPC1RAB9AHPGDSMN1; SMN2MAPT
SCHEMBL200799 0.83 LTA4H (0.46) LTA4HHPGDMAPK14SMN1; SMN2MAPT
SCHEMBL20836088 0.75 LIPE (0.43) LTA4HNPC1RAB9APPARGSMN1; SMN2
SCHEMBL202753 0.75 PARP10 (0.53) LTA4HSMN1; SMN2PARP10SRD5A2ERCC5
SCHEMBL22071794 0.73 MMP13 (0.47) NPC1RAB9AHPGDMAPK14SMN1; SMN2
SCHEMBL1730420 0.72 SMN1; SMN2 (0.66) NPC1RAB9AHPGDCRHBPCRHR2
SCHEMBL3739816 0.72 LTA4H (0.53) LTA4HNPC1RAB9AHPGDCRHBP
SCHEMBL4480029 0.72 PARP10 (0.55) LTA4HSMN1; SMN2ALDH1A1KMT2APARP10
SCHEMBL15588847 0.72 PARP10 (0.46) LTA4HSMN1; SMN2PARP10SRD5A2ERCC5
SCHEMBL454784 0.72 PARP10 (0.42) LTA4HNPC1RAB9ASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016170545-A1 PROCESS FOR THE PREPARATION OF 1-[(3R)-3-[4-AMINO-3-(4-PHENOXYPHENVL)-1H- PVRAZOLO[3,4-D]PYRINIIDIN-1-Y1]-1-PIPERIDINVL]-2-PROPEN-1-ONE AND ITS POLYMORPHS THEREOF MSN LABORATORIES PRIVATE LIMITED (IN) 2016-10-27 WO disclosed