SCHEMBL1817443

SCHEMBL1817443

CC1(C)OB(c2ccc3nc(Cl)cnc3c2)OC1(C)C

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
EGFR P00533 2/20 0.43
LPL P06858 9/20 0.39
LIPG Q9Y5X9 9/20 0.39
SNCA P37840 1/20 0.38
IRAK4 Q9NWZ3 1/20 0.38
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
ALPL P05186 1/20 0.34
AAK1 Q2M2I8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1814466 0.94 ALDH1A1 (0.44) ALDH1A1EGFRLPLLIPGSNCA
SCHEMBL21176048 0.82 LPL (0.39) EGFRLPLLIPGSNCAIRAK4
SCHEMBL18171891 0.81 EGFR (0.40) EGFRLPLLIPGSNCAIRAK4
SCHEMBL20622695 0.80 LPL (0.45) EGFRLPLLIPGSNCAIRAK4
SCHEMBL7603285 0.80 LPL (0.47) ALDH1A1LPLLIPGSNCA
SCHEMBL24145964 0.79 EGFR (0.46) EGFRLPLLIPGSNCAIRAK4
SCHEMBL14721612 0.79 EGFR (0.43) EGFRLPLLIPGSNCAIRAK4
SCHEMBL18614454 0.79 LPL (0.37) EGFRLPLLIPGSNCAIRAK4
SCHEMBL933108 0.79 LPL (0.44) EGFRLPLLIPGSNCAIRAK4
SCHEMBL31503579 0.78 TLR9 (0.52) ALDH1A1LPLLIPG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2321296-A1 SUBSTITUTED 5-AMINOPYRAZOLES AND USE THEREOF Bayer Schering Pharma Aktiengesellschaft (DE) 2011-05-18 EP disclosed
WO-2010020363-A1 SUBSTITUTED 5-AMINOPYRAZOLES AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-02-25 WO disclosed