SCHEMBL18175072

SCHEMBL18175072

CC(=O)Cn1cnc2c1COCN2C

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.36
PDE4B Q07343 2/20 0.36
PDE4C Q08493 2/20 0.36
PDE4D Q08499 2/20 0.36
ADORA2B P29275 2/20 0.36
ADORA2A P29274 1/20 0.36
TRPA1 O75762 1/20 0.33
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
KDM4E B2RXH2 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
POLB P06746 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15384288 0.87 TRPA1 (0.37) TRPA1KDM4E
SCHEMBL18175106 0.68 NPC1 (0.50) NPC1KDM4EPOLB
SCHEMBL12878629 0.59 NPC1 (0.50) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL17192909 0.58 POLB (0.36) SMN1; SMN2POLB
SCHEMBL10881570 0.57 KDM4E (0.65) NPC1KDM4ESMN1; SMN2POLB
SCHEMBL11531219 0.57 ADORA2B (0.78) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL16374759 0.57 MEN1 (0.42) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL15493510 0.56 CSNK2A1 (0.73) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL11983579 0.56 NPC1 (0.59) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL22521924 0.56 ALDH1A1 (0.46) ADORA2BKDM4ESMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170309-B1 2,6-DIOXO,-2,3-DIHYDRO-1H-PURINE COMPOUNDS USEFUL FOR TREATING DISORDERS RELATED TO THE ACTIVITY OF THE TRPA1 CHANNEL HYDRA BIOSCIENCES INC (US) 2016-10-26 EP disclosed