SCHEMBL18175810

SCHEMBL18175810

COc1cccc(CNC(=O)I)c1

nearest known ligand 0.74

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.68
MMP13 P45452 3/20 0.68
HTT P42858 1/20 0.68
SMN1; SMN2 Q16637 1/20 0.68
HPGD P15428 3/20 0.62
POLB P06746 1/20 0.62
EPHX2 P34913 2/20 0.60
LMNA P02545 2/20 0.60
KDM4E B2RXH2 1/20 0.60
USP2 O75604 1/20 0.60
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60
APEX1 P27695 1/20 0.59
RAB9A P51151 1/20 0.58
GAA P10253 1/20 0.58
MAPT P10636 1/20 0.58
ALOX15 P16050 1/20 0.58
GFER P55789 1/20 0.58
HSD17B10 Q99714 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3815151 0.87 ALDH1A1 (0.72) ALDH1A1MMP13HTTSMN1; SMN2HPGD
SCHEMBL660541 0.85 MMP13 (0.70) ALDH1A1MMP13HTTSMN1; SMN2HPGD
SCHEMBL2931410 0.85 MMP13 (0.70) ALDH1A1MMP13HTTSMN1; SMN2HPGD
SCHEMBL8245692 0.84 ALDH1A1 (0.68) ALDH1A1MMP13HTTSMN1; SMN2HPGD
Hydrochloric Acid SCHEMBL29194804 0.84 MMP13 (0.68) ALDH1A1MMP13HTTSMN1; SMN2HPGD
SCHEMBL30104666 0.84 ALDH1A1 (0.68) ALDH1A1MMP13HTTSMN1; SMN2HPGD
SCHEMBL13853495 0.83 ALDH1A1 (0.67) ALDH1A1MMP13HTTSMN1; SMN2HPGD
SCHEMBL934348 0.83 ALDH1A1 (0.76) ALDH1A1MMP13HTTSMN1; SMN2HPGD
SCHEMBL23771131 0.81 ALDH1A1 (0.65) ALDH1A1MMP13HTTSMN1; SMN2HPGD
SCHEMBL15471187 0.81 MMP13 (0.65) ALDH1A1MMP13HTTSMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616469-B1 9H-PURINE COMPOUNDS AS PI3K-DELTA INHIBITORS AND METHODS FOR THEIR MANUFACTURE EXELIXIS INC (US) 2016-10-26 EP disclosed