SCHEMBL18184641

SCHEMBL18184641

O=C(Cc1ccccn1)N1CCCCN2CC[C@@H]2C1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PAX8 Q06710 2/20 0.49
ALDH1A1 P00352 4/20 0.44
KDM4E B2RXH2 2/20 0.44
CNR1 P21554 1/20 0.44
L3MBTL3 Q96JM7 3/20 0.44
L3MBTL1 Q9Y468 3/20 0.44
MAPK1 P28482 1/20 0.43
ATM Q13315 1/20 0.43
TP53BP1 Q12888 1/20 0.43
HRH3 Q9Y5N1 4/20 0.42
EPHX2 P34913 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10574538 0.81 ALDH1A1 (0.58) PAX8ALDH1A1KDM4ECNR1L3MBTL1
SCHEMBL18184487 0.79 PAX8 (0.55) PAX8ALDH1A1KDM4ECNR1MAPK1
SCHEMBL4498993 0.79 ALDH1A1 (0.53) PAX8ALDH1A1KDM4ECNR1L3MBTL1
SCHEMBL18184488 0.76 PAX8 (0.50) PAX8ALDH1A1KDM4ECNR1MAPK1
SCHEMBL6037163 0.72 KDM4E (0.70) ALDH1A1KDM4ECNR1MAPK1EPHX2
SCHEMBL10572949 0.72 ALDH1A1 (0.56) ALDH1A1KDM4ECNR1L3MBTL1EPHX2
SCHEMBL30793971 0.72 KDM4E (0.54) PAX8ALDH1A1KDM4ECNR1L3MBTL1
SCHEMBL13826420 0.72 EPHX2 (0.54) ALDH1A1KDM4ECNR1HRH3EPHX2
SCHEMBL2603243 0.71 KDM4E (0.50) ALDH1A1KDM4ECNR1L3MBTL1EPHX2
SCHEMBL16002869 0.71 EPHX2 (0.56) ALDH1A1KDM4ECNR1L3MBTL1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016172631-A2 SUBSTRATE SELECTIVE INHIBITORS OF INSULIN-DEGRADING ENZYME (IDE) AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2016-10-27 WO disclosed