SCHEMBL18196844

SCHEMBL18196844

c1c[nH]c(CCCNCCNC23CC4CC(CC(C4)C2)C3)c1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 7/20 0.36
EPHX1 P07099 1/20 0.36
EPHX2 P34913 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
BCHE P06276 1/20 0.35
ACHE P22303 1/20 0.35
ADRB2 P07550 1/20 0.33
ADRB1 P08588 1/20 0.33
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18196906 0.85 HTR1A (0.38) HTR1AEPHX2BCHEACHEADRB2
SCHEMBL15013195 0.78 KDM4E (0.44) HTR1AEPHX2ADRB2ADRB1KDM4E
SCHEMBL1779571 0.78 EPHX1 (0.58) EPHX1EPHX2NPC1RAB9AALDH1A1
SCHEMBL18190630 0.76 HTR1A (0.41) HTR1AEPHX2NPC1RAB9AADRB2
SCHEMBL18190570 0.69 HTR1A (0.41) HTR1ANPC1RAB9AADRB2ADRB1
SCHEMBL3362927 0.68 EPHX2 (0.63) EPHX1EPHX2NPC1RAB9AALDH1A1
SCHEMBL3188537 0.67 GRIN2D (0.50) EPHX1EPHX2
SCHEMBL27647894 0.66 P2RX7 (0.36) EPHX2
SCHEMBL7003873 0.65 GPR84 (0.41)
SCHEMBL19914464 0.65 MEN1 (0.47) HTR1AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016176450-A1 TAMBJAMINES AND B-RING FUNCTIONALIZED PRODIGININES PORTLAND STATE UNIVERSITY (US) 2016-11-03 WO disclosed