SCHEMBL18199057

SCHEMBL18199057

C=C1NCCc2cc(C(C)(C)C)ccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 10/20 0.40
PARP1 P09874 5/20 0.40
PARP11 Q9NR21 5/20 0.39
HTR1D P28221 3/20 0.36
ADRA1A P35348 3/20 0.36
ADRA2A P08913 2/20 0.36
ADRA2B P18089 2/20 0.36
ADRA2C P18825 2/20 0.36
ADRA1D P25100 2/20 0.36
HTR1B P28222 2/20 0.36
ADRA1B P35368 2/20 0.36
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 1/20 0.35
PLA2G1B P04054 1/20 0.35
NFKB1 P19838 1/20 0.35
CASP3 P42574 1/20 0.35
RAB9A P51151 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
SENP8 Q96LD8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13186636 0.84 PARP10 (0.36) PARP10PARP1PARP11
SCHEMBL1432009 0.80 PARP10 (0.63) PARP10PARP1PARP11F7F3
SCHEMBL20024355 0.78 ALDH1A1 (0.47) ALDH1A1NPC1PLA2G1BNFKB1CASP3
SCHEMBL13186621 0.77 PARP10 (0.32) PARP10PARP1PARP11HSD17B10
SCHEMBL25733035 0.77 ALDH1A1 (0.40) ALDH1A1NPC1PLA2G1BNFKB1CASP3
SCHEMBL10100725 0.75 DRD2 (0.53) PARP10PARP1HTR1DADRA1AADRA2A
SCHEMBL13760475 0.74 DRD2 (0.56) PARP10PARP1PARP11F7F3
SCHEMBL19142931 0.74 CASP1 (0.47) PARP10PARP1PARP11ALDH1A1NPC1
SCHEMBL18199094 0.74 PARP10 (0.54) PARP10PARP1PARP11NISCH
SCHEMBL13512608 0.74 PARP10 (0.64) PARP10PARP1PARP11F7F3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2403846-B1 INHIBITORS OF BRUTON'S TYROSINE KINASE HOFFMANN LA ROCHE (CH) 2016-11-02 EP disclosed