SCHEMBL18214768

SCHEMBL18214768

Cc1nc(C(C)(O)C(F)(F)F)co1

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ENPP3 O14638 1/20 0.32
ENPP1 P22413 1/20 0.32
HSD11B1 P28845 3/20 0.31
AR P10275 1/20 0.31
NR1H2 P55055 1/20 0.31
NR1H3 Q13133 1/20 0.31
PTGS2 P35354 1/20 0.31
TLR7 Q9NYK1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18214769 0.82 ENPP3 (0.32) ENPP3ENPP1NR1H2NR1H3PTGS2
SCHEMBL18214733 0.79 ENPP3 (0.35) ENPP3ENPP1
SCHEMBL16996969 0.78 ENPP3 (0.34) ENPP3ENPP1PTGS2
SCHEMBL9911978 0.77 PTGS2 (0.40) ENPP3ENPP1PTGS2TLR7
SCHEMBL29131216 0.76 ENPP3 (0.34) ENPP3ENPP1PTGS2
SCHEMBL2656541 0.74 ENPP3 (0.42) ENPP3ENPP1
SCHEMBL23320613 0.73 ENPP3 (0.32) ENPP3ENPP1PTGS2TLR7
SCHEMBL18867386 0.71 ENPP3 (0.35) ENPP3ENPP1
SCHEMBL18214835 0.71 ENPP3 (0.32) ENPP3ENPP1
SCHEMBL20462629 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016177686-A1 PYRIDAZINE DERIVATIVES AS RORc MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2016-11-10 WO disclosed