SCHEMBL18215445

SCHEMBL18215445

O=C1N[C@@H](C(C(=O)O)C(=O)O)c2ccc(Br)cc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 2/20 0.44
EDNRA P25101 2/20 0.44
BCL2 P10415 1/20 0.37
MCL1 Q07820 1/20 0.37
CYP1A2 P05177 1/20 0.36
MAPK1 P28482 1/20 0.36
TGM2 P21980 1/20 0.36
CES1 P23141 1/20 0.36
CCNB2 O95067 1/20 0.35
CDK1 P06493 1/20 0.35
HSP90AA1 P07900 1/20 0.35
CCNB1 P14635 1/20 0.35
CCR6 P51684 1/20 0.35
CCNB3 Q8WWL7 1/20 0.35
S100A4 P26447 1/20 0.34
PTPRC P08575 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
NQO2 P16083 1/20 0.33
CA1 P00915 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18209302 1.00 EDNRB (0.44) EDNRBEDNRABCL2MCL1CYP1A2
SCHEMBL18209300 0.85 EDNRB (0.42) EDNRBEDNRABCL2MCL1CYP1A2
SCHEMBL18215457 0.83 TDP2 (0.38) EDNRBEDNRABCL2MCL1CYP1A2
SCHEMBL18209326 0.83 TDP2 (0.38) EDNRBEDNRABCL2MCL1CYP1A2
SCHEMBL23784644 0.82 TGM2 (0.36) TGM2CES1TDP2TP53MDM2
SCHEMBL18209303 0.78 HSD17B10 (0.51) EDNRBEDNRACYP1A2PARP1
SCHEMBL18215417 0.78 HSD17B10 (0.51) EDNRBEDNRACYP1A2PARP1
SCHEMBL18209306 0.76 HSD17B10 (0.47) EDNRBEDNRACYP1A2MAPK1TGM2
SCHEMBL18215447 0.76 HSD17B10 (0.47) EDNRBEDNRACYP1A2MAPK1TGM2
SCHEMBL23784662 0.72 TDP2 (0.35) EDNRBEDNRABCL2HSP90AA1NQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3292102-B1 ISOINDOLINONES, PROCESSES FOR THE PRODUCTION OF CHIRAL DERIVATIVES THEREOF AND USE THEREOF UNIV DEGLI STUDI DI SALERNO (IT) 2021-09-08 EP disclosed
WO-2016178140-A1 ISOINDOLINONES, PROCESSES FOR THE PRODUCTION OF CHIRAL DERIVATIVES THEREOF AND USE THEREOF UNIVERSITA' DEGLI STUDI DI SALERNO (IT) 2016-11-10 WO disclosed