SCHEMBL1821585

SCHEMBL1821585

CC(C)CCNC(=O)c1cnc(Cl)nc1C(F)(F)F

nearest known ligand 0.57

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 14/20 0.57
ATF1 P18846 13/20 0.57
XPO1 O14980 4/20 0.54
JUN P05412 2/20 0.53
NFKB2 Q00653 2/20 0.53
RELA Q04206 2/20 0.53
LMNA P02545 1/20 0.47
SCD O00767 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7489466 0.86 NFKB1 (0.59) NFKB1ATF1XPO1JUNNFKB2
SCHEMBL2307377 0.83 NFKB1 (0.61) NFKB1ATF1XPO1JUNNFKB2
SCHEMBL6977551 0.80 NFKB1 (0.62) NFKB1ATF1XPO1JUNNFKB2
SCHEMBL1822766 0.77 ATF1 (0.46) NFKB1ATF1LMNASCD
SCHEMBL4745582 0.75 CNR2 (0.69) NFKB1ATF1XPO1LMNA
SCHEMBL3379524 0.74 CNR2 (0.64) NFKB1ATF1XPO1
SCHEMBL3380681 0.74 CNR2 (0.64) NFKB1ATF1XPO1
SCHEMBL6288528 0.74 ATF1 (0.68) NFKB1ATF1XPO1JUNNFKB2
SCHEMBL8518174 0.73 NFKB1 (0.62) NFKB1ATF1XPO1JUNNFKB2
SCHEMBL3378920 0.73 CNR2 (0.64) NFKB1ATF1XPO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8030488-B2 Piperazine derivatives as stearoyl-coa desaturase inhibitors and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2011-10-04 US disclosed
EP-2316828-A1 Piperazine derivatives and their use as therapeutic agents Xenon Pharmaceuticals Inc. (CA) 2011-05-04 EP disclosed