SCHEMBL18229447

SCHEMBL18229447

O=C(Cc1c[nH]c2ccccc12)Nc1ccccc1Br

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.57
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
STAT3 P40763 1/20 0.57
RAB9A P51151 1/20 0.57
HSD17B10 Q99714 1/20 0.57
EGFR P00533 1/20 0.56
ERBB2 P04626 1/20 0.56
GLA P06280 1/20 0.56
MAPK8 P45983 1/20 0.55
LMNA P02545 2/20 0.54
ALDH1A1 P00352 2/20 0.54
CYP1A2 P05177 1/20 0.54
POLB P06746 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 1/20 0.54
PKM P14618 1/20 0.54
HTT P42858 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28373298 0.85 GLA (0.56) MAPTMEN1KMT2ASTAT3RAB9A
SCHEMBL28369557 0.85 MAPT (0.58) MAPTMEN1KMT2ASTAT3RAB9A
SCHEMBL18229452 0.84 CTSL (0.62) MAPTMEN1KMT2ASTAT3RAB9A
SCHEMBL28373392 0.84 MAPT (0.59) MAPTMEN1KMT2ASTAT3RAB9A
SCHEMBL28373046 0.84 LMNA (0.68) MAPTMEN1KMT2ASTAT3RAB9A
SCHEMBL9205145 0.83 KMT2A (0.62) MAPTMEN1KMT2ASTAT3RAB9A
SCHEMBL1519724 0.81 MAPT (0.64) MAPTMEN1KMT2ASTAT3RAB9A
SCHEMBL28619019 0.81 MAPK8 (0.55) MAPTMEN1KMT2ASTAT3RAB9A
SCHEMBL28341452 0.81 MAPT (0.75) MAPTMEN1KMT2ASTAT3RAB9A
SCHEMBL28167969 0.81 MAPT (0.69) MAPTMEN1KMT2ASTAT3RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016181414-A1 PROCESS FOR THE SYNTHESIS OF IVACAFTOR AND RELATED COMPOUNDS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2016-11-17 WO claimed
CN-107149602-B Application of indole compounds and derivatives thereof in preparation of anti-HIV drugs 中国医学科学院药物研究所 2020-10-09 CN disclosed
CN-107149603-B Application of indole compounds and derivatives thereof in preparation of anti-influenza virus drugs 中国医学科学院药物研究所 2020-07-14 CN disclosed
CN-107176921-B Indole compounds with antiviral activity in isatis root and derivatives thereof 中国医学科学院药物研究所 2020-03-31 CN disclosed
WO-2016181414-A1 PROCESS FOR THE SYNTHESIS OF IVACAFTOR AND RELATED COMPOUNDS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2016-11-17 WO disclosed