SCHEMBL18236296

SCHEMBL18236296

Ic1nc(-c2ccccn2)c(-c2ccccn2)s1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 7/20 0.49
KDM4E B2RXH2 6/20 0.47
NPC1 O15118 3/20 0.47
MAPT P10636 2/20 0.47
RAB9A P51151 2/20 0.47
GLA P06280 1/20 0.47
LMNA P02545 2/20 0.45
CCR1 P32246 2/20 0.45
CCR5 P51681 2/20 0.45
CCR8 P51685 2/20 0.45
CYP1A2 P05177 1/20 0.45
POLB P06746 1/20 0.45
METAP1 P53582 1/20 0.45
BLM P54132 1/20 0.45
HIF1A Q16665 1/20 0.45
DOHH Q9BU89 1/20 0.45
P4HTM Q9NXG6 1/20 0.45
ATM Q13315 1/20 0.44
TDP1 Q9NUW8 2/20 0.44
TP53 P04637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650294 0.71 KDM4E (0.51) TGFBR1KDM4ENPC1MAPTRAB9A
SCHEMBL323086 0.71 KDM4E (0.68) KDM4ENPC1MAPTRAB9AGLA
SCHEMBL6743757 0.70 KDM4E (0.60) KDM4ENPC1MAPTRAB9AGLA
Dipyridyl SCHEMBL2386179 0.68 KDM4E (0.93) KDM4ENPC1MAPTRAB9AGLA
Dipyridyl SCHEMBL8514685 0.68 KDM4E (0.93) KDM4ENPC1MAPTRAB9AGLA
Dipyridyl SCHEMBL31663992 0.68 KDM4E (0.93) KDM4ENPC1MAPTRAB9AGLA
SCHEMBL21495007 0.68 TGFBR1 (0.63) TGFBR1MAPTCYP1A2
SCHEMBL4614666 0.67 KDM4E (0.54) KDM4ENPC1MAPTRAB9AGLA
SCHEMBL6744657 0.67 KDM4E (0.56) KDM4ENPC1MAPTRAB9AGLA
SCHEMBL176039 0.67 KDM4E (0.68) KDM4ENPC1MAPTRAB9AGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016183173-A1 ANTIPARASITIC COMPOUNDS Avista Pharma Solutions (US) 2016-11-17 WO disclosed