SCHEMBL18239642

SCHEMBL18239642

Cc1cc(OC(F)(F)F)cc2cc[nH]c12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.34
TAF1 P21675 1/20 0.34
BRPF1 P55201 1/20 0.34
CREBBP Q92793 1/20 0.34
CECR2 Q9BXF3 1/20 0.34
BRD9 Q9H8M2 1/20 0.34
POLB P06746 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
PDE10A Q9Y233 2/20 0.34
GPR3 P46089 2/20 0.33
FFAR4 Q5NUL3 1/20 0.33
ABL1 P00519 1/20 0.33
BCR P11274 1/20 0.33
KDM4E B2RXH2 1/20 0.33
SCN8A Q9UQD0 3/20 0.32
SCN10A Q9Y5Y9 3/20 0.32
PTGS1 P23219 3/20 0.32
PTGS2 P35354 3/20 0.32
HRH4 Q9H3N8 1/20 0.32
KAT2B Q92831 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30644862 1.00 BRD4 (0.34) BRD4TAF1BRPF1CREBBPCECR2
SCHEMBL5372057 0.79 MEN1 (0.47) POLBMEN1MAPK1KMT2A
SCHEMBL7930189 0.78 HTR1A (0.36) BRD4TAF1BRPF1CREBBPCECR2
SCHEMBL18299637 0.77 PDE2A (0.32) BRD4TAF1BRPF1CREBBPCECR2
SCHEMBL18299986 0.75 KIF11 (0.38) BRD4TAF1BRPF1CREBBPCECR2
SCHEMBL18298885 0.73 KIF11 (0.41) POLBGPR3FFAR4ABL1BCR
SCHEMBL30039737 0.73 KIF11 (0.41) POLBGPR3FFAR4ABL1BCR
SCHEMBL4484912 0.72 AHR (0.47) BRD4TAF1BRPF1CREBBPCECR2
SCHEMBL18300000 0.71 MTNR1A (0.35) PDE10AGPR3FFAR4KDM4EPTGS1
Pivalate SCHEMBL30711319 0.71 KMT2A (0.38) POLBKDM4EPTGS1MEN1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 41 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250230127-A1 MONO- OR DI-SUBSTITUTED INDOLE DERIVATIVES AS DENGUE VIRAL REPLICATION INHIBITORS JANSSEN PHARMACEUTICALS INC (US) 2025-07-17 US disclosed
US-12172959-B2 Mono- or di-substituted indole derivatives as dengue viral replication inhibitors Janssen Pharmaceuticals, Inc. (US) 2024-12-24 US disclosed
US-20240182414-A1 MONO- OR DI-SUBSTITUTED INDOLE DERIVATIVES AS DENGUE VIRAL REPLICATION INHIBITORS Janssen Pharmaceuticals, Inc. (US) 2024-06-06 US disclosed
US-11827602-B2 Mono- or di-substituted indole derivatives as dengue viral replication inhibitors Janssen Pharmaceuticals, Inc. (US) 2023-11-28 US disclosed
US-11827602-B2 Mono- or di-substituted indole derivatives as dengue viral replication inhibitors Janssen Pharmaceuticals, Inc. (US) 2023-11-28 US disclosed
US-20230066771-A1 NUCLEAR RECEPTOR MODULATORS ABBVIE INC (US) 2023-03-02 US disclosed
US-20230066771-A1 NUCLEAR RECEPTOR MODULATORS ABBVIE INC (US) 2023-03-02 US disclosed
EP-3896072-B1 MONO- OR DI-SUBSTITUTED INDOLE DERIVATIVES AS DENGUE VIRAL REPLICATION INHIBITORS JANSSEN PHARMACEUTICALS INC (US) 2022-11-16 EP disclosed
EP-3896072-B1 MONO- OR DI-SUBSTITUTED INDOLE DERIVATIVES AS DENGUE VIRAL REPLICATION INHIBITORS JANSSEN PHARMACEUTICALS INC (US) 2022-11-16 EP disclosed
EP-3896072-A1 MONO- OR DI-SUBSTITUTED INDOLE DERIVATIVES AS DENGUE VIRAL REPLICATION INHIBITORS Janssen Pharmaceuticals, Inc. (US) 2021-10-20 EP disclosed
CN-107820494-A Nuclear receptor modulators 艾伯维公司 2018-03-20 CN disclosed
WO-2017167950-A1 SUBSTITUTED INDOLE DERIVATIVES AS DENGUE VIRAL REPLICATION INHIBITORS Janssen Pharmaceuticals, Inc. (US) 2017-10-05 WO disclosed
WO-2017046258-A1 MONO- OR DI-SUBSTITUTED INDOLE DERIVATIVES AS DENGUE VIRAL REPLICATION INHIBITORS Janssen Pharmaceuticals, Inc. (US) 2017-03-23 WO disclosed
WO-2017046255-A1 MONO- OR DI-SUBSTITUTED INDOLE DERIVATIVES AS DENGUE VIRAL REPLICATION INHIBITORS Janssen Pharmaceuticals, Inc. (US) 2017-03-23 WO disclosed
WO-2016200851-A1 NUCLEAR RECEPTOR MODULATORS ABBVIE INC. (US) 2016-12-15 WO disclosed
WO-2016200851-A1 NUCLEAR RECEPTOR MODULATORS ABBVIE INC. (US) 2016-12-15 WO disclosed
US-20160362370-A1 NUCLEAR RECEPTOR MODULATORS ABBVIE INC. (US) 2016-12-15 US disclosed
US-20160362370-A1 NUCLEAR RECEPTOR MODULATORS ABBVIE INC. (US) 2016-12-15 US disclosed
US-20160362370-A1 NUCLEAR RECEPTOR MODULATORS ABBVIE INC. (US) 2016-12-15 US disclosed
WO-2016180696-A1 MONO- OR DI-SUBSTITUTED INDOLE DERIVATIVES AS DENGUE VIRAL REPLICATION INHIBITORS Janssen Pharmaceuticals, Inc. (US) 2016-11-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160362370-A1 NUCLEAR RECEPTOR MODULATORS NR1I2, NR1H2, NR5A2 BRD4 758/4885TAF1 897/4885BRPF1 1191/4885
US-20250230127-A1 MONO- OR DI-SUBSTITUTED INDOLE DERIVATIVES AS DENGUE VIRAL REPLICATION INHIBITORS IDO1, IDO2, IRF3 BRD4 358/4885TAF1 4100/4885BRPF1 2721/4885
US-11827602-B2 Mono- or di-substituted indole derivatives as dengue viral replication inhibitors IDO1, IDO2, IRF3 BRD4 346/4885TAF1 4064/4885BRPF1 2616/4885
US-20240182414-A1 MONO- OR DI-SUBSTITUTED INDOLE DERIVATIVES AS DENGUE VIRAL REPLICATION INHIBITORS IDO1, IDO2, IRF3 BRD4 346/4885TAF1 4064/4885BRPF1 2616/4885
US-12172959-B2 Mono- or di-substituted indole derivatives as dengue viral replication inhibitors IDO1, IDO2, IRF3 BRD4 346/4885TAF1 4064/4885BRPF1 2616/4885
US-20230066771-A1 NUCLEAR RECEPTOR MODULATORS NR1I2, NR1H2, NR5A2 BRD4 758/4885TAF1 897/4885BRPF1 1191/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.