SCHEMBL18239882

SCHEMBL18239882

CCCCOc1cc2c(c(C(=O)CCl)c1)OCC(=O)N2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.43
ALDH1A1 P00352 2/20 0.43
RXFP1 Q9HBX9 1/20 0.41
NR3C2 P08235 1/20 0.39
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
ADRB2 P07550 5/20 0.38
ADRB1 P08588 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.36
DRD2 P14416 3/20 0.36
HTR2A P28223 2/20 0.36
DRD1 P21728 1/20 0.36
DRD4 P21917 1/20 0.36
DRD5 P21918 1/20 0.36
DRD3 P35462 1/20 0.36
MAOA P21397 2/20 0.36
MAOB P27338 2/20 0.36
HTR1A P08908 2/20 0.35
SLC6A4 P31645 1/20 0.35
CRBN Q96SW2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12428840 0.89 MAPT (0.41) MAPTALDH1A1RXFP1NR3C2PDE3B
SCHEMBL12428824 0.87 NR3C2 (0.43) MAPTALDH1A1RXFP1NR3C2PDE3B
SCHEMBL18239918 0.83 MAPT (0.37) MAPTALDH1A1RXFP1NR3C2PDE3B
SCHEMBL561100 0.81 MAOA (0.46) MAPTALDH1A1ADRB2ADRB1SMN1; SMN2
SCHEMBL30223645 0.81 MAOA (0.46) MAPTALDH1A1ADRB2ADRB1SMN1; SMN2
SCHEMBL17484547 0.76 ADRB2 (0.39) MAPTALDH1A1RXFP1ADRB2ADRB1
SCHEMBL12428821 0.76 ADRB2 (0.48) ADRB2ADRB1HTR2AHTR1ASLC6A4
SCHEMBL12648407 0.75 DRD2 (0.40) MAPTRXFP1NR3C2PDE3BPDE3A
SCHEMBL20285626 0.72 NR3C2 (0.38) MAPTALDH1A1RXFP1NR3C2PDE3B
SCHEMBL17476304 0.71 SMYD3 (0.56) MAPTALDH1A1DRD2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016180349-A1 BIPHENYL DERIVATIVE HAVING BETA2 RECEPTOR EXCITEMENT AND M RECEPTOR ANTAGONISTIC ACTIVITIES AND APPLICATION THEREFOF IN MEDICAMENT 四川海思科制药有限公司 2016-11-17 WO disclosed