SCHEMBL1825481

SCHEMBL1825481

Fc1cc(Cl)ccc1C1CCNC1

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 0.54
CHRNB2 P17787 1/20 0.49
CHRNA4 P43681 1/20 0.49
SLC6A2 P23975 2/20 0.45
SLC6A4 P31645 2/20 0.45
SLC6A3 Q01959 2/20 0.45
OPRL1 P41146 2/20 0.44
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
HTR2B P41595 1/20 0.43
CHRM1 P11229 1/20 0.43
CHRM3 P20309 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29904538 1.00 HTR3A (0.54) HTR3ACHRNB2CHRNA4SLC6A2SLC6A4
SCHEMBL16455075 0.90 HTR3A (0.47) HTR3ACHRNB2CHRNA4SLC6A2SLC6A4
SCHEMBL29932045 0.90 SLC6A2 (0.51) HTR3ACHRNB2CHRNA4SLC6A2SLC6A4
SCHEMBL3385011 0.90 SLC6A2 (0.51) HTR3ACHRNB2CHRNA4SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL16446414 0.89 HTR3A (0.46) HTR3ACHRNB2CHRNA4SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL29931941 0.88 SLC6A2 (0.50) HTR3ASLC6A2SLC6A4SLC6A3OPRL1
Hydrochloric Acid SCHEMBL4890844 0.88 SLC6A2 (0.50) HTR3ASLC6A2SLC6A4SLC6A3OPRL1
SCHEMBL1822160 0.83 CHRNB2 (0.51) CHRNB2CHRNA4SLC6A2SLC6A4SLC6A3
SCHEMBL29904548 0.83 CHRNB2 (0.51) CHRNB2CHRNA4SLC6A2SLC6A4SLC6A3
SCHEMBL20438926 0.83 CHRNB2 (0.51) CHRNB2CHRNA4SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250109148-A1 HETEROCYCLIC GLP-1 AGONISTS SHANGHAI SHOUTI BIOTECHNOLOGY CO., LTD. (CN) 2025-04-03 US disclosed
EP-2155669-B1 NEW DISUBSTITUTED PHENYLPYRROLIDINES AS MODULATORS OF CORTICAL CATECHOLAMINERGIC NEUROTRANSMISSION NSAB AF NEUROSEARCH SWEDEN AB (DK) 2011-05-04 EP disclosed
US-20100197760-A1 DISUBSTITUTED PHENYLPYRROLIDINES AS MODULATORS OF CORTICAL CATECHOLAMINERGIC NEUROTRANSMISSION NSAB, FILIAL AF NEUROSEARCH SWEDEN AB, SVERIGE (DK) 2010-08-05 US disclosed
CN-101711234-A New disubstituted phenylpyrrolidines as modulators of cortical catecholaminergic neurotransmission NSAB OF NEUROSEARCH SWEDEN AB 2010-05-19 CN disclosed
EP-2155669-A1 NEW DISUBSTITUTED PHENYLPYRROLIDINES AS MODULATORS OF CORTICAL CATECHOLAMINERGIC NEUROTRANSMISSION NSAB, Filial af NeuroSearch Sweden AB, Sverige (DK) 2010-02-24 EP disclosed
WO-2008148799-A1 NEW DISUBSTITUTED PHENYLPYRROLIDINES AS MODULATORS OF CORTICAL CATECHOLAMINERGIC NEUROTRANSMISSION NSAB, FILIAL OF NEUROSEARCH SWEDEN AB, SVERIGE (DK) 2008-12-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250109148-A1 HETEROCYCLIC GLP-1 AGONISTS GLP1R, GIPR, GCGR HTR3A 138/4885CHRNB2 1212/4885CHRNA4 1328/4885
US-20100197760-A1 DISUBSTITUTED PHENYLPYRROLIDINES AS MODULATORS OF CORTICAL CATECHOLAMINERGIC NEUROTRANSMISSION SLC6A2, SLC6A3, SLC18A2 HTR3A 53/4885CHRNB2 33/4885CHRNA4 18/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.