SCHEMBL18258134

SCHEMBL18258134

CCn1c(N)cc2ccc(OC)c(OC)c21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.37
NQO2 P16083 1/20 0.37
GAA P10253 4/20 0.36
KDM4E B2RXH2 4/20 0.35
MAPT P10636 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
HSD17B10 Q99714 3/20 0.34
HTT P42858 1/20 0.34
ALDH1A1 P00352 2/20 0.33
KMT2A Q03164 2/20 0.33
PTGS2 P35354 1/20 0.33
TUBB4A P04350 1/20 0.33
TUBB P07437 1/20 0.33
TUBA3C P0DPH7 1/20 0.33
TUBA1B P68363 1/20 0.33
TUBA4A P68366 1/20 0.33
TUBB4B P68371 1/20 0.33
TUBB3 Q13509 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21335595 0.84 CYP19A1 (0.42) CYP19A1NQO2GAAKDM4EMAPT
SCHEMBL18247727 0.78 CYP19A1 (0.40) CYP19A1NQO2GAAMAPTALDH1A1
SCHEMBL18247494 0.69 TUBB4A (0.44) CYP19A1NQO2GAAKDM4EMAPT
SCHEMBL29953247 0.62 CYP19A1 (0.43) CYP19A1NQO2KDM4EMAPTNPSR1
SCHEMBL1742563 0.62 KDM4E (0.46) CYP19A1NQO2GAAKDM4EMAPT
SCHEMBL21335586 0.62 CCR2 (0.43) CYP19A1NQO2GAAKDM4EMAPT
SCHEMBL27199552 0.61 TDP1 (0.46) KDM4ESMN1; SMN2HSD17B10HTTKMT2A
SCHEMBL30498072 0.61 TDP1 (0.46) KDM4ESMN1; SMN2HSD17B10HTTKMT2A
SCHEMBL30701949 0.61 CA9 (0.50) CYP19A1KDM4EMAPTSMN1; SMN2ALDH1A1
SCHEMBL3674074 0.61 CA9 (0.50) CYP19A1KDM4EMAPTSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016185279-A1 BENZOIMIDAZOLE DERIVATIVES AS PAD4 INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2016-11-24 WO disclosed