SCHEMBL18266293

SCHEMBL18266293

CCC(=O)Nc1cc(C(=O)NCc2ccc(COCC(F)(F)I)cc2)cc(C)n1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.38
ADORA3 P0DMS8 4/20 0.37
ADORA1 P30542 3/20 0.37
EPHX2 P34913 2/20 0.36
NR1H4 Q96RI1 1/20 0.36
ADORA2A P29274 1/20 0.36
MAPT P10636 3/20 0.36
ALDH1A1 P00352 2/20 0.35
GAA P10253 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
PPARG P37231 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
KDM4E B2RXH2 1/20 0.35
PKM P14618 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2715325 0.92 ALDH1A1 (0.44) SCN9AADORA3ADORA1EPHX2ADORA2A
SCHEMBL18266371 0.90 SCN9A (0.39) SCN9AEPHX2NR1H4MAPTALDH1A1
SCHEMBL18266731 0.88 SCN9A (0.48) SCN9AADORA3EPHX2NR1H4MAPT
SCHEMBL2716263 0.82 EPHX2 (0.54) SCN9AEPHX2NR1H4ALDH1A1GAA
SCHEMBL2717517 0.82 ALDH1A1 (0.46) SCN9AEPHX2NR1H4MAPTALDH1A1
SCHEMBL2713229 0.81 EPHX2 (0.54) SCN9AADORA3ADORA1EPHX2NR1H4
SCHEMBL2714168 0.80 SCN9A (0.51) SCN9AEPHX2MAPTALDH1A1MEN1
SCHEMBL18266145 0.79 WDR5 (0.40) SCN9AADORA3ADORA1ADORA2AMEN1
SCHEMBL18266380 0.79 KMT2A (0.47) ADORA3ADORA1ADORA2AGAAMEN1
SCHEMBL2717677 0.79 PTGES (0.45) SCN9AEPHX2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2630122-B1 ARYLAMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC (JP) 2016-11-30 EP disclosed