SCHEMBL18266554

SCHEMBL18266554

Cc1cc(C(=O)NCc2cc(C)c(OCC(C)F)c(C)c2)cc(NC(=O)C(C)(C)O)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.39
CCR3 P51677 2/20 0.33
NR1H4 Q96RI1 1/20 0.32
ALDH1A1 P00352 2/20 0.32
RET P07949 2/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
CHRNB2 P17787 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
CHRNA4 P43681 1/20 0.31
TP53 P04637 1/20 0.31
MAPT P10636 1/20 0.31
GAA P10253 1/20 0.31
MMP13 P45452 1/20 0.30
PTGES O14684 1/20 0.30
MAP4K1 Q92918 1/20 0.30
CHRM4 P08173 2/20 0.30
USP2 O75604 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2716526 0.94 SCN9A (0.38) SCN9ACCR3NR1H4ALDH1A1RET
SCHEMBL2714698 0.82 SCN9A (0.48) SCN9ACCR3ALDH1A1KDM4EMEN1
SCHEMBL2714301 0.82 PTGES (0.40) SCN9ACCR3NR1H4ALDH1A1MMP13
SCHEMBL2713499 0.82 SCN9A (0.38) SCN9ACCR3ALDH1A1KDM4EMEN1
SCHEMBL2717877 0.81 CHRNB2 (0.37) SCN9ACCR3ALDH1A1RETKDM4E
SCHEMBL2714754 0.80 SCN9A (0.37) SCN9AALDH1A1MEN1KMT2ACHRNB2
SCHEMBL2716387 0.78 SCN9A (0.41) SCN9ACCR3ALDH1A1KMT2AMAPT
SCHEMBL2716573 0.77 PPARG (0.41) NR1H4
SCHEMBL18266581 0.77 LMNA (0.41)
SCHEMBL2717500 0.77 PPARG (0.40) SCN9ANR1H4ALDH1A1MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2630122-B1 ARYLAMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC (JP) 2016-11-30 EP disclosed