SCHEMBL18266802

SCHEMBL18266802

Cc1cc(C(=O)NCc2ccc(OC(F)(F)I)c(Cl)c2)cc(NC(=O)C(C)C)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 4/20 0.52
ROCK2 O75116 1/20 0.41
SCN3A Q9NY46 6/20 0.41
WDR5 P61964 3/20 0.40
LMNA P02545 1/20 0.40
SCN1A P35498 2/20 0.38
SCN5A Q14524 2/20 0.38
SCN2A Q99250 2/20 0.38
SCN8A Q9UQD0 2/20 0.38
SCN10A Q9Y5Y9 2/20 0.38
KCNH2 Q12809 1/20 0.38
KCNB1 Q14721 1/20 0.38
GAA P10253 1/20 0.38
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
MAPT P10636 1/20 0.37
PKM P14618 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CCR3 P51677 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2716384 0.93 SCN9A (0.53) SCN9AROCK2SCN3AWDR5LMNA
SCHEMBL2715174 0.85 SCN9A (0.51) SCN9AWDR5LMNAKCNH2KCNB1
SCHEMBL2714516 0.84 SCN9A (0.49) SCN9AROCK2WDR5KCNB1PPARD
SCHEMBL2713199 0.83 SCN9A (0.48) SCN9AROCK2SCN3AKCNB1
SCHEMBL2715099 0.83 SCN9A (0.56) SCN9AROCK2SCN3ACCR3
SCHEMBL2714086 0.83 ROCK2 (0.50) SCN9AROCK2SCN3AWDR5LMNA
SCHEMBL2715396 0.81 SCN9A (0.48) SCN9AROCK2SCN3AKCNB1PTGES
SCHEMBL2714916 0.81 EPHX2 (0.53) SCN9AKCNB1GAAKDM4ESMN1; SMN2
SCHEMBL2719098 0.80 SCN9A (0.51) SCN9AKCNB1MAPTPTGESPPARD
SCHEMBL18266303 0.80 SCN9A (0.47) SCN9AROCK2LMNAKCNB1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2630122-B1 ARYLAMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC (JP) 2016-11-30 EP disclosed