SCHEMBL18270779

SCHEMBL18270779

O=C(O)c1cc2c(Cl)c(F)ccc2s1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.48
CCNC P24863 1/20 0.44
CDK8 P49336 1/20 0.44
DAO P14920 3/20 0.43
BCKDK O14874 2/20 0.43
BCL2L1 Q07817 2/20 0.42
GPR35 Q9HC97 2/20 0.42
MCL1 Q07820 3/20 0.41
RXFP1 Q9HBX9 1/20 0.41
PLK4 O00444 2/20 0.41
AURKA O14965 2/20 0.41
DAPK3 O43293 2/20 0.41
CHEK2 O96017 2/20 0.41
CDK1 P06493 2/20 0.41
PIM1 P11309 2/20 0.41
CDK2 P24941 2/20 0.41
MAPK9 P45984 2/20 0.41
CSNK1D P48730 2/20 0.41
GSK3A P49840 2/20 0.41
GSK3B P49841 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15697576 0.83 HDAC3 (0.49) NOTUMCCNCCDK8DAOBCKDK
SCHEMBL30714157 0.80 GPR35 (0.42) NOTUMCCNCCDK8DAOBCL2L1
SCHEMBL26111219 0.80 GPR35 (0.42) NOTUMCCNCCDK8DAOBCL2L1
SCHEMBL4805937 0.80 STING1 (0.43) CCNCCDK8BCL2L1GPR35PLK4
SCHEMBL18264006 0.79 HDAC3 (0.43) RXFP1HDAC3HDAC4HDAC1HDAC6
SCHEMBL2893037 0.77 SLC9A1 (0.62) NOTUMBCL2L1GPR35PLK4AURKA
SCHEMBL17858538 0.73 CHRNA7 (0.49) NOTUMDAOBCKDKBCL2L1GPR35
SCHEMBL9262314 0.73 ALDH1A1 (0.46) NOTUMCCNCCDK8DAOBCKDK
SCHEMBL1853420 0.73 DAO (0.46) NOTUMCCNCCDK8DAOBCKDK
SCHEMBL18264120 0.73 DAO (0.46) NOTUMCCNCCDK8DAOBCKDK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016191366-A1 MODULATORS FOR NICOTINIC ACETYLCHOLINE RECEPTOR α2 AND α4 SUBUNITS THE SCRIPPS RESEARCH INSTITUTE (US) 2016-12-01 WO disclosed