SCHEMBL1827596

SCHEMBL1827596

CCSC1=NC2(C[C@](CC)(c3ccccc3)Oc3ccc(Br)cc32)C(=O)N1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 5/20 0.37
CTSD P07339 2/20 0.37
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
DYRK3 O43781 1/20 0.32
PIM1 P11309 1/20 0.32
CSNK2A2 P19784 1/20 0.32
CSNK2B P67870 1/20 0.32
CSNK2A1 P68400 1/20 0.32
DYRK1A Q13627 1/20 0.32
CSNK2A3 Q8NEV1 1/20 0.32
DYRK2 Q92630 1/20 0.32
DYRK1B Q9Y463 1/20 0.32
TP53 P04637 1/20 0.31
MEN1 O00255 2/20 0.30
KMT2A Q03164 2/20 0.30
LMNA P02545 1/20 0.30
ALPL P05186 1/20 0.30
HSP90AA1 P07900 1/20 0.30
ALPI P09923 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3244223 0.88 KDM4E (0.33) DYRK3PIM1CSNK2A2CSNK2BCSNK2A1
SCHEMBL1830168 0.85 BACE1 (0.43) BACE1CTSDOPRM1OPRD1TP53
SCHEMBL1828675 0.83 BACE1 (0.34) BACE1CTSDTP53
SCHEMBL1828991 0.78 BACE1 (0.42) BACE1CTSDOPRM1OPRD1TP53
SCHEMBL1827435 0.75 BACE1 (0.40) BACE1CTSDOPRM1OPRD1TP53
SCHEMBL1828383 0.74 BACE1 (0.39) BACE1CTSDOPRM1OPRD1MEN1
SCHEMBL1826421 0.70 BACE1 (0.47) BACE1CTSDOPRM1OPRD1
SCHEMBL1831618 0.69 BACE1 (0.39) BACE1CTSD
SCHEMBL3241071 0.68 BACE1 (0.39) BACE1CTSDTP53MEN1KMT2A
SCHEMBL1827904 0.67 BACE1 (0.40) BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2324032-A2 INHIBITORS OF BETA-SECRETASE Vitae Pharmaceuticals, Inc. (US) 2011-05-25 EP disclosed
WO-2010021680-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-02-25 WO disclosed