SCHEMBL3244223

SCHEMBL3244223

CCSC1=NC2(CC(CC)(c3ccccc3)Oc3ccccc32)C(=O)N1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.33
TSHR P16473 3/20 0.32
MEN1 O00255 2/20 0.32
CYP1A2 P05177 2/20 0.32
KMT2A Q03164 2/20 0.32
POLB P06746 1/20 0.32
APEX1 P27695 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
CYP2D6 P10635 2/20 0.31
CYP2C19 P33261 2/20 0.31
PKM P14618 1/20 0.31
NFKB1 P19838 1/20 0.31
THPO P40225 1/20 0.31
ADRA2A P08913 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NISCH Q9Y2I1 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1827596 0.88 BACE1 (0.37) KDM4EMEN1KMT2ALMNADYRK3
SCHEMBL1830168 0.72 BACE1 (0.43) HSD11B1
SCHEMBL1822743 0.72 CYP2D6 (0.30) TSHRMEN1CYP1A2KMT2ACYP2D6
SCHEMBL1828675 0.71 BACE1 (0.34)
SCHEMBL1828991 0.65 BACE1 (0.42) MEN1KMT2AHSD11B1
SCHEMBL9378722 0.63 BACE1 (0.43) CYP3A4
SCHEMBL11009062 0.63 KDM4E (0.39) KDM4ETSHRMEN1CYP1A2KMT2A
SCHEMBL27281924 0.61 SIGMAR1 (0.45) TSHRMEN1CYP1A2KMT2ACYP2D6
SCHEMBL6837134 0.61 ESR1 (0.36) TSHRMEN1CYP1A2KMT2ATDP1
SCHEMBL9182623 0.57 HCAR3 (0.42) TSHRMEN1CYP1A2KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010021680-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-02-25 WO disclosed