SCHEMBL182828

SCHEMBL182828

c1ccc(OCCN2CCC(N3CCCC3)CC2)cc1

nearest known ligand 0.84

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 7/20 0.72
LTA4H P09960 10/20 0.63
TMEM97 Q5BJF2 1/20 0.61
SIGMAR1 Q99720 1/20 0.61
CHRM1 P11229 1/20 0.55
DRD2 P14416 1/20 0.55
KCNH2 Q12809 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL182574 0.85 HRH3 (0.69) HRH3LTA4H
SCHEMBL255201 0.84 LTA4H (0.86) HRH3LTA4H
Ammonia Solution, Strong SCHEMBL264615 0.82 LTA4H (0.83) HRH3LTA4H
SCHEMBL5870409 0.82 LTA4H (0.83) HRH3LTA4HKCNH2
SCHEMBL3951411 0.82 LTA4H (0.83) HRH3LTA4HKCNH2
SCHEMBL5943693 0.82 HRH3 (0.60) HRH3LTA4HKCNH2
SCHEMBL8109834 0.81 TMEM97 (0.68) HRH3LTA4HTMEM97SIGMAR1
SCHEMBL6943925 0.81 TMEM97 (0.68) HRH3LTA4HTMEM97SIGMAR1
SCHEMBL8693762 0.81 TMEM97 (0.68) LTA4HTMEM97SIGMAR1
Bromide SCHEMBL4827747 0.80 LTA4H (0.81) HRH3LTA4HKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049502-B1 2,4-SUBSTITUTED QUINAZOLINES AS LIPID KINASE INHIBITORS NOVARTIS AG (CH) 2012-01-04 EP disclosed