SCHEMBL18284227

SCHEMBL18284227

c1ccc(COc2ccc3ccn(Cc4ccc5ccccc5c4)c3c2)cc1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.59
HTR7 P34969 1/20 0.55
MAPK14 Q16539 1/20 0.52
CYP3A4 P08684 1/20 0.47
HTR6 P50406 2/20 0.46
MCHR1 Q99705 1/20 0.45
KMT2A Q03164 2/20 0.44
BCL2 P10415 1/20 0.44
MCL1 Q07820 1/20 0.44
RAB9A P51151 2/20 0.44
NPC1 O15118 2/20 0.44
MEN1 O00255 1/20 0.44
MRGPRX4 Q96LA9 1/20 0.44
MAPT P10636 1/20 0.43
PTGER3 P43115 1/20 0.43
PTGDR Q13258 1/20 0.43
APP P05067 1/20 0.43
SNCA P37840 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6100496 0.91 ALOX5 (0.61) ALOX5HTR7MAPK14CYP3A4KMT2A
SCHEMBL6086767 0.88 MAPK14 (0.54) ALOX5HTR7MAPK14HTR6MCHR1
SCHEMBL6192092 0.83 HTR6 (0.59) ALOX5MAPK14HTR6KMT2ARAB9A
SCHEMBL3193186 0.81 MAPK14 (0.61) ALOX5MAPK14KMT2ARAB9ANPC1
SCHEMBL28349833 0.81 HDAC6 (0.65) MAPK14BCL2MCL1NPC1MAPT
SCHEMBL24414699 0.80 MAOB (0.56) ALOX5HTR7MAPK14HTR6MCHR1
SCHEMBL30991821 0.80 MAOB (0.56) ALOX5HTR7MAPK14HTR6MCHR1
SCHEMBL19172461 0.80 HTR7 (0.65) ALOX5HTR7MAPK14CYP3A4MCHR1
SCHEMBL6085680 0.80 HTR6 (0.65) HTR6KMT2A
SCHEMBL9208196 0.79 ALOX5 (0.48) ALOX5MAPK14HTR6KMT2ABCL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016196890-A1 INHIBITORS OF HEXOKINASE AND METHODS OF USE THEREOF VTV THERAPEUTICS LLC (US) 2016-12-08 WO disclosed