SCHEMBL1828535

SCHEMBL1828535

NC(=O)Oc1[nH]c2ccc(CN3CCCC(C(N)=O)C3)cc2c1Sc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.47
LTA4H P09960 1/20 0.44
ICAM1 P05362 1/20 0.42
LMNA P02545 2/20 0.41
KMT2A Q03164 2/20 0.40
ATM Q13315 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
MBTPS1 Q14703 1/20 0.39
MAPT P10636 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
POLB P06746 1/20 0.39
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
MEN1 O00255 1/20 0.38
ROCK2 O75116 1/20 0.38
CCR2 P41597 1/20 0.38
ROCK1 Q13464 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1824155 0.88 KDM4E (0.42) KMT2ACYP2C9KDM4EALDH1A1HPGD
SCHEMBL1616243 0.87 GAA (0.49) GAALTA4HICAM1LMNAKMT2A
SCHEMBL1823764 0.83 GAA (0.39) GAALTA4HKMT2AMAPTKDM4E
SCHEMBL1824756 0.83 CXCR4 (0.41) KMT2AKDM4EALDH1A1HPGDMEN1
SCHEMBL1825695 0.82 PARP1 (0.44) GAALMNAL3MBTL1MAPTKDM4E
SCHEMBL1823170 0.82 SPHK2 (0.43)
SCHEMBL1823810 0.79 ALDH1A1 (0.43) GAALMNAKMT2ACYP3A4NPSR1
SCHEMBL1826204 0.79 MCHR2 (0.38) KMT2AMAPTKDM4EALDH1A1HPGD
SCHEMBL1821784 0.78 FAAH (0.37) MAPTKDM4EALDH1A1HPGD
SCHEMBL1826566 0.78 DRD4 (0.44) GAALMNAL3MBTL1MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1794122-B1 3-SUBSTITUTED-5- AND 6-AMINOALKYL INDOLE-2-CARBOXYLIC ACID AMIDES AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE I AVENTIS PHARMA INC (US) 2011-05-04 EP claimed