SCHEMBL18288652

SCHEMBL18288652

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nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 4/20 0.45
ESR1 P03372 1/20 0.35
POLB P06746 1/20 0.35
ESR2 Q92731 1/20 0.35
CTDSP1 Q9GZU7 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
KEAP1 Q14145 1/20 0.35
NFE2L2 Q16236 1/20 0.35
CA12 O43570 1/20 0.32
AKR1B10 O60218 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
AKR1B1 P15121 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32
CA14 Q9ULX7 1/20 0.32
CHRNB2 P17787 2/20 0.31
CHRNA4 P43681 2/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18288691 1.00 HCAR2 (0.45) HCAR2ESR1POLBESR2CTDSP1
SCHEMBL2609714 0.92 HCAR2 (0.50) HCAR2ESR1POLBESR2CTDSP1
SCHEMBL2115988 0.92 HCAR2 (0.59) HCAR2ESR1POLBESR2CTDSP1
SCHEMBL2115986 0.92 HCAR2 (0.59) HCAR2ESR1POLBESR2CTDSP1
SCHEMBL18288707 0.80 HCAR2 (0.43) HCAR2KEAP1NFE2L2CA12AKR1B10
SCHEMBL18288684 0.78 HCAR2 (0.42) HCAR2KEAP1NFE2L2CA12AKR1B10
SCHEMBL18288690 0.77 ALDH1A1 (0.50) HCAR2KEAP1NFE2L2
SCHEMBL18288701 0.77 ALDH1A1 (0.50) HCAR2KEAP1NFE2L2
SCHEMBL2172419 0.76 TSHR (0.48) ESR1POLBESR2CTDSP1TDP1
SCHEMBL18288682 0.74 HCAR2 (0.38) HCAR2TDP1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160355464-A1 FUMARATE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND METHODS OF USE Nguyen, Mark Quang (US) 2016-12-08 US disclosed
US-20160355464-A1 FUMARATE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND METHODS OF USE Nguyen, Mark Quang (US) 2016-12-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160355464-A1 FUMARATE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND METHODS OF USE FH, FPGS, APC HCAR2 290/4885ESR1 3585/4885POLB 471/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.