SCHEMBL1829600

SCHEMBL1829600

COCCCOc1cccc(B2OC(C)(C)C(C)(C)O2)c1.COCCCOc1cccc(Br)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.48
LPL P06858 1/20 0.43
LIPG Q9Y5X9 1/20 0.43
ALDH1A1 P00352 3/20 0.41
MAPT P10636 1/20 0.41
KMT2A Q03164 1/20 0.41
LMNA P02545 1/20 0.40
FFAR1 O14842 1/20 0.39
PPARG P37231 1/20 0.39
PPARD Q03181 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MAOB P27338 6/20 0.38
NOS1 P29475 1/20 0.38
HMOX2 P30519 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1830523 0.94 LPL (0.48) KDM4ELPLLIPGALDH1A1CYP1A2
SCHEMBL31150275 0.91 LPL (0.48) KDM4ELPLLIPGALDH1A1CYP1A2
SCHEMBL431636 0.87 LIPG (0.46) KDM4ELPLLIPGALDH1A1CYP1A2
SCHEMBL2801619 0.84 LPL (0.51) LPLLIPGALDH1A1MAOB
SCHEMBL18124821 0.84 LIPG (0.50) LPLLIPGMAPK1
SCHEMBL20745594 0.83 LPL (0.43) KDM4ELPLLIPGALDH1A1LMNA
Cyclopentane SCHEMBL28665515 0.83 LPL (0.43) KDM4ELPLLIPGALDH1A1CYP1A2
SCHEMBL8445213 0.83 LPL (0.48) LPLLIPGMAOB
SCHEMBL1821482 0.82 KDM4E (0.63) KDM4EALDH1A1MAPTKMT2ALMNA
SCHEMBL4602862 0.81 LPL (0.49) LPLLIPGKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2324032-A2 INHIBITORS OF BETA-SECRETASE Vitae Pharmaceuticals, Inc. (US) 2011-05-25 EP disclosed
WO-2010021680-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-02-25 WO disclosed