SCHEMBL18306103

SCHEMBL18306103

CN1C[C@@H](C(=O)O)OC1=O

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACE P12821 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
MAPT P10636 1/20 0.32
POLB P06746 4/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
BRD4 O60885 2/20 0.32
CYP2C9 P11712 1/20 0.31
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10249510 1.00 ACE (0.34) ACESMN1; SMN2MAPTPOLBL3MBTL1
SCHEMBL18305954 1.00 ACE (0.34) ACESMN1; SMN2MAPTPOLBL3MBTL1
SCHEMBL22772528 0.82 MAOA (0.40)
SCHEMBL22300991 0.79 BRD4 (0.47) BRD4
SCHEMBL10284517 0.75 CYP2C9 (0.34) SMN1; SMN2POLBL3MBTL1CYP2C9GAA
SCHEMBL8294508 0.73 L3MBTL1 (0.49) ACEPOLBL3MBTL1
SCHEMBL3271191 0.72 L3MBTL1 (0.45) POLBL3MBTL1CYP2C9GAA
SCHEMBL16869473 0.72 CYP3A4 (0.38) ACEMAPTPOLBBRD4GAA
SCHEMBL9057946 0.71
SCHEMBL925260 0.71 SIRT1 (0.48) SMN1; SMN2POLBL3MBTL1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3307741-A1 POSITIVE ALLOSTERIC MODULATORS OF MUSCARINIC M2 RECEPTOR Bayer Pharma Aktiengesellschaft (DE) 2018-04-18 EP disclosed
WO-2016198342-A1 POSITIVE ALLOSTERIC MODULATORS OF MUSCARINIC M2 RECEPTOR BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-12-15 WO disclosed