SCHEMBL18308366

SCHEMBL18308366

COC(=O)c1c(OC)cc2c(C)n[nH]c2c1N

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.38
POLB P06746 1/20 0.38
ALDH1A1 P00352 4/20 0.38
HPGD P15428 3/20 0.38
GAA P10253 3/20 0.38
NPSR1 Q6W5P4 2/20 0.38
GABRA1 P14867 1/20 0.37
GABRA5 P31644 1/20 0.37
GABRA3 P34903 1/20 0.37
GABRA2 P47869 1/20 0.37
GABRA6 Q16445 1/20 0.37
MAPT P10636 4/20 0.37
MAPK1 P28482 2/20 0.37
HSD17B10 Q99714 2/20 0.37
TDP1 Q9NUW8 1/20 0.36
CISD2 Q8N5K1 1/20 0.36
CSNK2A2 P19784 1/20 0.35
KDR P35968 1/20 0.35
CSNK2B P67870 1/20 0.35
CSNK2A1 P68400 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4077018 0.78 NQO2 (0.38) KDM4EALDH1A1HPGDGAAGABRA1
SCHEMBL18306146 0.75 ADORA2A (0.49) KDM4EPOLBALDH1A1HPGDNPSR1
SCHEMBL8532411 0.69 KDM4E (0.45) KDM4EPOLBALDH1A1HPGDGAA
SCHEMBL4403769 0.69 LMNA (0.49) ALDH1A1HPGDKMT2AHTTLMNA
SCHEMBL1144821 0.69 CNR2 (0.49) KDM4EHPGDMAPK1KMT2AHTT
SCHEMBL26046787 0.68 POLB (0.45) KDM4EPOLBALDH1A1HPGDGAA
SCHEMBL1144834 0.68 HSD17B2 (0.49) KDM4EALDH1A1HPGDGAANPSR1
SCHEMBL14384290 0.67 KDM4E (0.53) KDM4EPOLBALDH1A1HPGDGAA
SCHEMBL1145139 0.67 AR (0.43) KDM4EPOLBALDH1A1HPGDGAA
SCHEMBL18308520 0.67 S100B (0.39) KDM4EPOLBALDH1A1HPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016199943-A1 HETEROCYCLIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-12-15 WO disclosed