SCHEMBL18322930

SCHEMBL18322930

CN1CCN(c2c(-c3ccc(OC4CCN(CCC=O)CC4)cc3)cnc3ccccc23)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SSTR2 P30874 3/20 0.43
HRH3 Q9Y5N1 6/20 0.41
RAB9A P51151 2/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
ADRA1A P35348 2/20 0.38
KCNH2 Q12809 2/20 0.38
CHRM4 P08173 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
MET P08581 1/20 0.37
MAP4K1 Q92918 1/20 0.37
SCN9A Q15858 1/20 0.36
BMPR1B O00238 1/20 0.36
BMPR1A P36894 1/20 0.36
ACVRL1 P37023 1/20 0.36
ACVR1 Q04771 1/20 0.36
HTR2A P28223 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18322893 0.90 SSTR2 (0.41) SSTR2HRH3ADRA1AKCNH2CHRM4
SCHEMBL18322921 0.86 HRH3 (0.42) SSTR2HRH3ADRA1AKCNH2MEN1
SCHEMBL18322980 0.84 HRH3 (0.42) HRH3ADRA1AKCNH2HTR2AHTR7
SCHEMBL18322841 0.84 HRH3 (0.42) HRH3RAB9ANPC1ADRA1AKCNH2
SCHEMBL18319018 0.82 SSTR2 (0.43) SSTR2HRH3RAB9ANPC1ALDH1A1
SCHEMBL18319044 0.77 NAMPT (0.51) SSTR2ALDH1A1KDM4E
SCHEMBL18319042 0.77 NAMPT (0.51) SSTR2ALDH1A1KDM4E
SCHEMBL18322938 0.76 CHRNB1 (0.43) HRH3ADRA1AKCNH2
SCHEMBL18318480 0.73 PIK3CD (0.44) SSTR2RAB9AALDH1A1SMN1; SMN2KCNH2
SCHEMBL18322895 0.72 HRH3 (0.40) HRH3ALDH1A1ADRA1AKCNH2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3310441-A1 1, 4-SUBSTITUTED PIPERIDINE DERIVATIVES Cephalon, Inc. (US) 2018-04-25 EP disclosed
WO-2016205633-A1 1, 4-SUBSTITUTED PIPERIDINE DERIVATIVES CEPHALON, INC. (US) 2016-12-22 WO disclosed