SCHEMBL18322982

SCHEMBL18322982

O=CCCN1CC[C@H](Oc2ccc(-c3ccc4cccnc4c3)cc2)C1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.43
PDE3B Q13370 2/20 0.42
PDE3A Q14432 2/20 0.42
PDE10A Q9Y233 2/20 0.42
ESR1 P03372 3/20 0.40
CHEK2 O96017 1/20 0.38
FASN P49327 3/20 0.37
DRD2 P14416 1/20 0.35
CHRM2 P08172 1/20 0.35
CHRM3 P20309 1/20 0.35
HTR7 P34969 1/20 0.35
HTR1A P08908 1/20 0.35
FDPS P14324 1/20 0.35
ROCK1 Q13464 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18322904 0.94 GSK3B (0.42) GSK3BPDE3BPDE3APDE10ACHEK2
SCHEMBL18322946 0.79 HTR7 (0.37) GSK3BCHEK2HTR7HTR1AROCK1
SCHEMBL18322979 0.78 GSK3B (0.42) GSK3BFASNDRD2HTR7
SCHEMBL18318608 0.77 PIK3CD (0.54) GSK3BPDE3BPDE3APDE10AFASN
SCHEMBL18318113 0.77 PIK3CD (0.54) GSK3BPDE3BPDE3APDE10AFASN
SCHEMBL18318114 0.77 PIK3CD (0.54) GSK3BPDE3BPDE3APDE10AFASN
SCHEMBL18322976 0.77 ROCK1 (0.39) HTR1AFDPSROCK1
SCHEMBL18322938 0.76 CHRNB1 (0.43) CHEK2FASN
Hydrochloric Acid SCHEMBL18318506 0.76 PIK3CD (0.53) GSK3BPDE3BPDE3APDE10AFASN
Hydrochloric Acid SCHEMBL18318626 0.76 PIK3CD (0.53) GSK3BPDE3BPDE3APDE10AFASN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3310441-A1 1, 4-SUBSTITUTED PIPERIDINE DERIVATIVES Cephalon, Inc. (US) 2018-04-25 EP disclosed
WO-2016205633-A1 1, 4-SUBSTITUTED PIPERIDINE DERIVATIVES CEPHALON, INC. (US) 2016-12-22 WO disclosed