SCHEMBL18323926

SCHEMBL18323926

Cc1ccc2c(c1)CNCN2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR5A P47898 3/20 0.39
PARP10 Q53GL7 2/20 0.37
PARP11 Q9NR21 1/20 0.37
ALDH1A1 P00352 2/20 0.34
GAA P10253 2/20 0.34
MAPT P10636 2/20 0.34
HSD17B10 Q99714 1/20 0.34
EPHX2 P34913 1/20 0.33
PARP1 P09874 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRNB2 P17787 1/20 0.32
CHRNA4 P43681 1/20 0.32
PNMT P11086 1/20 0.31
CYP1A2 P05177 3/20 0.31
CYP2C19 P33261 2/20 0.31
NPC1 O15118 1/20 0.31
CYP2C9 P11712 1/20 0.31
RAB9A P51151 1/20 0.31
MCL1 Q07820 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14294948 0.83 HTR5A (0.43) HTR5APARP10PARP11ALDH1A1GAA
SCHEMBL19257866 0.83
SCHEMBL19657741 0.82 GAA (0.41) HTR5APARP10PARP11ALDH1A1GAA
SCHEMBL290721 0.76 PNMT (0.48) PARP10PARP11PNMT
SCHEMBL7420026 0.76 MAPT (0.34) ALDH1A1GAAMAPTHSD17B10CHRNB2
SCHEMBL12545829 0.76 CHRNB2 (0.38) ALDH1A1GAAHSD17B10CHRNB2CHRNA4
SCHEMBL28590347 0.73 PARP10 (0.42) HTR5APARP10PARP11ALDH1A1GAA
SCHEMBL22093074 0.72 CYP2A6 (0.37) ALDH1A1GAAMAPTHSD17B10RAB9A
SCHEMBL4060436 0.72 PNMT (0.54) CHRNB2CHRNA4PNMT
SCHEMBL30020921 0.72 MAPT (0.44) HTR5APARP10PARP11ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2922840-B1 BICYCLIC HETEROCYCLE SUBSTITUTED PYRIDYL COMPOUNDS USEFUL AS KINASE MODULATORS BRISTOL MYERS SQUIBB CO (US) 2016-12-21 EP disclosed