SCHEMBL18338409

SCHEMBL18338409

Ic1cnn2c1NCCC2

nearest known ligand 0.30

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 1/20 0.30
CDK9 P50750 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1800727 0.77 CCNT1 (0.30) CCNT1CDK9
SCHEMBL7925552 0.77 MAPT (0.35) CCNT1CDK9
SCHEMBL17869465 0.77 CHRNB2 (0.31) CCNT1CDK9
SCHEMBL12265082 0.77 SSTR4 (0.32) CCNT1CDK9
Hydrochloric Acid SCHEMBL8156603 0.76
SCHEMBL4206342 0.73 DRD2 (0.33) CCNT1CDK9
SCHEMBL5151795 0.73 CYP11B1 (0.38)
SCHEMBL18013173 0.73 MAPT (0.36) CCNT1CDK9
SCHEMBL9869341 0.72 POLB (0.38) CCNT1CDK9
SCHEMBL25274344 0.70 CCNT1 (0.32) CCNT1CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240067655-A1 KINASE MODULATORS AND METHODS OF USE THEREOF NEURON23, INC. 2024-02-29 US disclosed
US-20220340592-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2022-10-27 US disclosed
US-11352369-B2 Pyridine and pyrimidine derivatives ASTRAZENECA AB (SE) 2022-06-07 US disclosed
US-11352369-B2 Pyridine and pyrimidine derivatives ASTRAZENECA AB (SE) 2022-06-07 US disclosed
EP-3539961-B1 POLYCYCLIC AMIDE DERIVATIVES AS CDK9 INHIBITORS ASTRAZENECA AB (SE) 2021-10-06 EP disclosed
EP-3539961-B1 POLYCYCLIC AMIDE DERIVATIVES AS CDK9 INHIBITORS ASTRAZENECA AB (SE) 2021-10-06 EP disclosed
US-20210171541-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2021-06-10 US disclosed
US-20210171541-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2021-06-10 US disclosed
CN-107873028-B Polycyclic amide derivatives useful as CDK9 inhibitors 阿斯利康(瑞典)有限公司 2021-02-02 CN disclosed
US-10717746-B2 Chemical compounds ASTRAZENECA AB (SE) 2020-07-21 US disclosed
EP-3539961-A1 POLYCYCLIC AMIDE DERIVATIVES AS CDK9 INHIBITORS Astrazeneca AB (SE) 2019-09-18 EP disclosed
EP-3539961-A1 POLYCYCLIC AMIDE DERIVATIVES AS CDK9 INHIBITORS Astrazeneca AB (SE) 2019-09-18 EP disclosed
EP-3313838-B1 POLYCYCLIC AMIDE DERIVATIVES AS CDK9 INHIBITORS ASTRAZENECA AB (SE) 2019-04-03 EP disclosed
EP-3313838-B1 POLYCYCLIC AMIDE DERIVATIVES AS CDK9 INHIBITORS ASTRAZENECA AB (SE) 2019-04-03 EP disclosed
US-20180093998-A1 CHEMICAL COMPOUNDS ASTRAZENECA PHARMACEUTICALS LP 2018-04-05 US disclosed
US-20180093998-A1 CHEMICAL COMPOUNDS ASTRAZENECA PHARMACEUTICALS LP 2018-04-05 US disclosed
US-9845331-B2 Chemical compounds ASTRAZENECA AB (SE) 2017-12-19 US disclosed
US-9845331-B2 Chemical compounds ASTRAZENECA AB (SE) 2017-12-19 US disclosed
WO-2017001354-A1 POLYCYCLIC AMIDE DERIVATIVES AS CDK9 INHIBITORS ASTRAZENECA AB (SE) 2017-01-05 WO disclosed
US-20160376287-A1 Chemical Compounds ASTRAZENECA AB (SE) 2016-12-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220340592-A1 CHEMICAL COMPOUNDS CDK9, BCL9, BCL9L CCNT1 49/4885CDK9 1/4885
US-20240067655-A1 KINASE MODULATORS AND METHODS OF USE THEREOF TYK2, NUAK1, NUAK2 CCNT1 3067/4885CDK9 289/4885
US-20210171541-A1 CHEMICAL COMPOUNDS CDK9, BCL9, BCL9L CCNT1 49/4885CDK9 1/4885
US-20160376287-A1 Chemical Compounds CDK9, BCL9, BCL9L CCNT1 49/4885CDK9 1/4885
US-10717746-B2 Chemical compounds CDK9, BCL9, BCL9L CCNT1 49/4885CDK9 1/4885
US-20180093998-A1 CHEMICAL COMPOUNDS CDK9, BCL9, BCL9L CCNT1 49/4885CDK9 1/4885
US-11352369-B2 Pyridine and pyrimidine derivatives CDK9, BCL9, CDK19 CCNT1 46/4885CDK9 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.