SCHEMBL1837239

SCHEMBL1837239

CSc1ncc(CC=O)c(NC(C)C)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 1/20 0.39
HTT P42858 2/20 0.34
ALDH1A1 P00352 2/20 0.33
SYK P43405 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
CDK1 P06493 1/20 0.32
CDK2 P24941 1/20 0.32
KDR P35968 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32
MAPT P10636 2/20 0.31
LMNA P02545 1/20 0.31
FOS P01100 1/20 0.31
JUN P05412 1/20 0.31
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30955646 0.82 AOC1 (0.40) TRPM8HTTALDH1A1SYKMEN1
SCHEMBL3968862 0.82 AOC1 (0.40) TRPM8HTTALDH1A1SYKMEN1
SCHEMBL1521487 0.82 TRPM8 (0.38) TRPM8HTTALDH1A1SYKMEN1
SCHEMBL1521541 0.82 HTT (0.48) TRPM8HTTALDH1A1SYKMEN1
SCHEMBL24170657 0.81 TRPM8 (0.37) TRPM8HTTALDH1A1SYKKDM4E
SCHEMBL25658788 0.81 TRPM8 (0.40) TRPM8HTTALDH1A1SYKMEN1
SCHEMBL5067063 0.80 MEN1 (0.34) TRPM8ALDH1A1SYKMEN1KMT2A
SCHEMBL24225121 0.79 HTT (0.39) TRPM8HTTALDH1A1SYKMEN1
SCHEMBL1841950 0.79 TRPM8 (0.41) TRPM8ALDH1A1MEN1KMT2ACDK1
SCHEMBL7504628 0.78 ALDH1A1 (0.40) ALDH1A1MEN1KMT2ATSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323986-A2 HETOEROCYCLYL CARBONIC ACID AMIDES AS ANTIPROLIFERATIVE AGENTS, PDKL INHIBITORS Boehringer Ingelheim International GmbH (DE) 2011-05-25 EP disclosed
EP-2321299-A2 PYRIDONS AS PDK1 INHIBITORS Boehringer Ingelheim International GmbH (DE) 2011-05-18 EP disclosed
WO-2010007114-A2 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-01-21 WO disclosed
WO-2010007116-A2 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-01-21 WO disclosed