SCHEMBL18375349

SCHEMBL18375349

CCc1cccc(-c2cnco2)c1C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.42
PKM P14618 1/20 0.42
IMPDH2 P12268 7/20 0.41
IMPDH1 P20839 3/20 0.41
AAK1 Q2M2I8 1/20 0.40
PDK2 Q15119 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
MAP4K4 O95819 1/20 0.38
ADRA1A P35348 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP19A1 P11511 1/20 0.38
EDNRB P24530 1/20 0.37
EDNRA P25101 1/20 0.37
PTK2 Q05397 1/20 0.37
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
P2RX7 Q99572 1/20 0.36
ADRA1D P25100 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24026537 0.80 IMPDH2 (0.43) IMPDH2IMPDH1AAK1CYP3A4CYP2D6
SCHEMBL18378811 0.80 LMNA (0.47) LMNAPKMIMPDH2IMPDH1PDK2
SCHEMBL18367723 0.75 LMNA (0.43) LMNAPKMIMPDH2IMPDH1AAK1
SCHEMBL28680769 0.75 ALDH1A1 (0.40) MEN1KMT2A
SCHEMBL19726598 0.74 LMNA (0.42) LMNAPKMIMPDH2IMPDH1PDK2
SCHEMBL26259988 0.73 MEN1 (0.48) LMNAPKMIMPDH2IMPDH1PDK2
SCHEMBL21163229 0.72 CYP1A2 (0.47) ADRA1ACYP2D6CYP19A1EDNRBEDNRA
SCHEMBL22150409 0.72 PDK2 (0.43) LMNAPKMIMPDH2IMPDH1AAK1
SCHEMBL16371219 0.70 IMPDH2 (0.60) IMPDH2IMPDH1AAK1MAP4K4CYP19A1
SCHEMBL27976182 0.70 AKR1B1 (0.44) LMNAPKMIMPDH2IMPDH1AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017007694-A1 6-AMINO-QUINOLINE-3-CARBONITRILS AS COT MODULATORS GILEAD SCIENCES, INC. (US) 2017-01-12 WO disclosed