Gsk-269962A

Gsk-269962A

SCHEMBL1838346

CCn1c(-c2nonc2N)nc2cnc(Oc3cccc(NC(=O)c4ccc(OCCN5CCOCC5)cc4)c3)cc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 10/20 1.00
AURKB Q96GD4 3/20 1.00
RPS6KA5 O75582 2/20 1.00
AURKA O14965 2/20 1.00
FLT3 P36888 2/20 1.00
CDC7 O00311 1/20 1.00
PLK4 O00444 1/20 1.00
DAPK3 O43293 1/20 1.00
ROCK2 O75116 1/20 1.00
PRKD3 O94806 1/20 1.00
PRKCG P05129 1/20 1.00
LCK P06239 1/20 1.00
PIM1 P11309 1/20 1.00
PRKACA P17612 1/20 1.00
RPS6KB1 P23443 1/20 1.00
CDK2 P24941 1/20 1.00
MARK3 P27448 1/20 1.00
AKT1 P31749 1/20 1.00
AKT2 P31751 1/20 1.00
FLT4 P35916 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Gsk-269962A SCHEMBL29365470 1.00 ROCK1 (1.00) ROCK1AURKBRPS6KA5AURKAFLT3
Gsk-269962A SCHEMBL29387396 1.00 ROCK1 (1.00) ROCK1AURKBRPS6KA5AURKAFLT3
Gsk-269962A SCHEMBL29715551 0.99 ROCK1 (0.99) ROCK1AURKBRPS6KA5AURKAFLT3
SCHEMBL4007749 0.95 ROCK1 (0.90) ROCK1AURKBRPS6KA5AURKAFLT3
SCHEMBL4002686 0.94 ROCK1 (0.89) ROCK1AURKBRPS6KA5AURKAFLT3
SCHEMBL4003195 0.94 ROCK1 (0.89) ROCK1AURKBRPS6KA5AURKAFLT3
SCHEMBL4002266 0.94 ROCK1 (0.88) ROCK1AURKBRPS6KA5AURKAFLT3
SCHEMBL4008685 0.93 ROCK1 (0.87) ROCK1AURKBRPS6KA5AURKAFLT3
SCHEMBL4004630 0.92 ROCK1 (0.85) ROCK1AURKBRPS6KA5AURKAFLT3
SCHEMBL4000210 0.91 ROCK1 (0.84) ROCK1AURKBRPS6KA5AURKAFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 137 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4692329-A1 COMPOSITION FOR INDUCING DIRECT DIFFERENTIATION OF STEM CELLS INTO CORNEAL ENDOTHELIAL CELLS AND METHOD FOR INDUCING DIRECT DIFFERENTIATION USING SAME The Asan Foundation (KR) 2026-02-11 EP claimed
EP-4636079-A1 METHOD FOR INDUCING DIFFERENTIATION OF STEM CELLS INTO CORNEAL ENDOTHELIAL CELLS AND USE THEREOF The Asan Foundation (KR) 2025-10-22 EP claimed
US-12371664-B2 Medium for direct differentiation of pluripotent stem cell-derived mesenchymal stem cell, method for preparing mesenchymal stem cell by using same, and mesenchymal stem cell prepared thereby CHA BIOTECH CO., LTD. (KR) 2025-07-29 US claimed
WO-2024210619-A1 COMPOSITION FOR INDUCING DIRECT DIFFERENTIATION OF STEM CELLS INTO CORNEAL ENDOTHELIAL CELLS AND METHOD FOR INDUCING DIRECT DIFFERENTIATION USING SAME 재단법인 아산사회복지재단 2024-10-10 WO claimed
WO-2024128696-A1 METHOD FOR INDUCING DIFFERENTIATION OF STEM CELLS INTO CORNEAL ENDOTHELIAL CELLS AND USE THEREOF 재단법인 아산사회복지재단 2024-06-20 WO claimed
US-20230391881-A1 COMPOSITIONS AND METHODS FOR OVERCOMING DR5-INDUCED IMMUNE EVASION BY SOLID TUMORS UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2023-12-07 US claimed
CN-106795487-B Method for proliferating pancreatic progenitor cells 武田药品工业株式会社 2021-11-19 CN claimed
US-20210340498-A1 MEDIUM FOR DIRECT DIFFERENTIATION OF PLURIPOTENT STEM CELL-DERIVED MESENCHYMAL STEM CELL, METHOD FOR PREPARING MESENCHYMAL STEM CELL BY USING SAME, AND MESENCHYMAL STEM CELL PREPARED THEREBY CHA BIOTECH CO., LTD. (KR) 2021-11-04 US claimed
EP-3848455-A1 MEDIUM FOR DIRECT DIFFERENTIATION OF PLURIPOTENT STEM CELL-DERIVED MESENCHYMAL STEM CELL, METHOD FOR PREPARING MESENCHYMAL STEM CELL BY USING SAME, AND MESENCHYMAL STEM CELL PREPARED THEREBY CHA Biotech Co., Ltd. (KR) 2021-07-14 EP claimed
US-10655105-B2 Method for proliferation of pancreatic progenitor cells TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2020-05-19 US claimed
US-7547779-B2 Preparation of 1,6-disubstituted azabenzimidazoles as kinase inhibitors GLAXO GROUP LIMITED (GB) 2009-06-16 US claimed
EP-1675552-A4 PREPERATION OF 1,6-DISUBSTITUTED AZABENZIMIDAZOLES AS KINASE INHIBITORS GLAXO GROUP LTD (GB) 2009-06-03 EP claimed
US-20080234261-A1 Preparation of 1,6-Disubstituted Azabenzimidazoles as Kinase Inhibitors GLAXOSMITHKLINE LLC 2008-09-25 US claimed
EP-1675552-A2 PREPERATION OF 1,6-DISUBSTITUTED AZABENZIMIDAZOLES AS KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-07-05 EP claimed
WO-2005037197-A2 PREPERATION OF 1,6-DISUBSTITUTED AZABENZIMIDAZOLES AS KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2005-04-28 WO claimed
US-20260062678-A1 CELL REPLACEMENT THERAPY FOR PULMONARY DISEASES THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2026-03-05 US disclosed
EP-4692329-A1 COMPOSITION FOR INDUCING DIRECT DIFFERENTIATION OF STEM CELLS INTO CORNEAL ENDOTHELIAL CELLS AND METHOD FOR INDUCING DIRECT DIFFERENTIATION USING SAME The Asan Foundation (KR) 2026-02-11 EP disclosed
EP-1675552-A2 PREPERATION OF 1,6-DISUBSTITUTED AZABENZIMIDAZOLES AS KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-07-05 EP disclosed
WO-2005037197-A2 PREPERATION OF 1,6-DISUBSTITUTED AZABENZIMIDAZOLES AS KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2005-04-28 WO disclosed
WO-2005037197-A2 PREPERATION OF 1,6-DISUBSTITUTED AZABENZIMIDAZOLES AS KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2005-04-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260062678-A1 CELL REPLACEMENT THERAPY FOR PULMONARY DISEASES WNT3A, BMP4, GSK3B ROCK1 12/4885AURKB 1983/4885RPS6KA5 774/4885
US-20230391881-A1 COMPOSITIONS AND METHODS FOR OVERCOMING DR5-INDUCED IMMUNE EVASION BY SOLID TUMORS CD274, PDCD1, PDCD1LG2 ROCK1 4/4885AURKB 416/4885RPS6KA5 1766/4885
US-20080234261-A1 Preparation of 1,6-Disubstituted Azabenzimidazoles as Kinase Inhibitors TNK2, ROCK1, ARHGDIB ROCK1 2/4885AURKB 101/4885RPS6KA5 99/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.