SCHEMBL1838732

SCHEMBL1838732

CCOC(=O)c1cccc(OCC(C2CCCCC2)C2(c3ccc(Cl)cc3)Nc3cc(F)c(F)cc3N2)n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 4/20 0.35
MGLL Q99685 1/20 0.35
CYP1A2 P05177 1/20 0.35
MDM4 O15151 3/20 0.35
MDM2 Q00987 2/20 0.35
TP53 P04637 2/20 0.35
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
MAPK1 P28482 1/20 0.33
ALDH1A1 P00352 1/20 0.32
CASP3 P42574 1/20 0.32
TLR4 O00206 1/20 0.32
TSHR P16473 1/20 0.32
P2RX3 P56373 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
KCNH2 Q12809 1/20 0.32
NR1H4 Q96RI1 1/20 0.32
PTGER1 P34995 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1839045 0.90 PTGER1 (0.35) CYP3A4CYP2C9NR1H4PTGER1
SCHEMBL1838536 0.84 SMN1; SMN2 (0.38) FAAHMGLLMDM4MDM2TP53
SCHEMBL1837083 0.83 GAA (0.39) FAAHTP53KMT2AALDH1A1KCNH2
SCHEMBL1840740 0.82 HCRTR1 (0.35) FAAHMGLLMDM4MDM2TP53
SCHEMBL1838605 0.81 ALOX15 (0.37) MDM2TP53MEN1KMT2AMAPK1
SCHEMBL1840527 0.80 ADRB3 (0.35) KMT2AALDH1A1KCNH2
SCHEMBL3236034 0.80 DRD4 (0.31)
SCHEMBL1841033 0.80 KDM4E (0.36) MEN1KMT2AALDH1A1CYP3A4CYP2D6
SCHEMBL1840570 0.79 NR1H4 (0.39) CYP3A4CYP2D6CYP2C9KCNH2NR1H4
SCHEMBL1839730 0.79 PPARA (0.41) FAAHCYP1A2MDM4MDM2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2321282-A1 NEW BENZIMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2011-05-18 EP disclosed
WO-2010028981-A1 NEW BENZIMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2010-03-18 WO disclosed