SCHEMBL18396554

SCHEMBL18396554

COC(=O)c1cccc([N+](=O)[O-])c1CC#N

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.54
MAPT P10636 2/20 0.54
MAPK1 P28482 2/20 0.54
KDM4E B2RXH2 3/20 0.53
PKM P14618 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
SMN1; SMN2 Q16637 3/20 0.47
HPGD P15428 1/20 0.47
TSHR P16473 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
POLB P06746 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
HSD17B10 Q99714 1/20 0.43
CTSD P07339 1/20 0.42
LMNA P02545 1/20 0.41
GLA P06280 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10192631 0.83 ALDH1A1 (0.58) ALDH1A1MAPTMAPK1KDM4EPKM
SCHEMBL27797486 0.82 ALDH1A1 (0.57) ALDH1A1MAPTMAPK1KDM4EPKM
SCHEMBL8113842 0.82 ALDH1A1 (0.57) ALDH1A1MAPTMAPK1KDM4EPKM
SCHEMBL332011 0.82 ALDH1A1 (0.57) ALDH1A1MAPTMAPK1KDM4EPKM
SCHEMBL17144681 0.81 ALDH1A1 (0.56) ALDH1A1MAPTMAPK1KDM4EPKM
SCHEMBL6655749 0.80 ALDH1A1 (0.53) ALDH1A1MAPTMAPK1KDM4EPKM
SCHEMBL528555 0.80 ALDH1A1 (0.58) ALDH1A1MAPTMAPK1KDM4EPKM
SCHEMBL20916593 0.80 ALDH1A1 (0.55) ALDH1A1MAPTMAPK1KDM4EPKM
SCHEMBL27431445 0.80 ALDH1A1 (0.55) ALDH1A1MAPTMAPK1KDM4EPKM
SCHEMBL11048095 0.80 ALDH1A1 (0.55) ALDH1A1MAPTMAPK1KDM4EPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017013593-A1 ISOQUINOLINONE DERIVATIVES AS PARP INHIBITORS LUPIN LIMITED (IN) 2017-01-26 WO disclosed
WO-2017013593-A1 ISOQUINOLINONE DERIVATIVES AS PARP INHIBITORS LUPIN LIMITED (IN) 2017-01-26 WO disclosed