SCHEMBL18399231

SCHEMBL18399231

CC(=O)n1ncc2cc(C)c(OC(=O)N3CCNCC3)cc21

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.40
AURKA O14965 1/20 0.40
DAPK3 O43293 1/20 0.40
CSNK1A1 P48729 1/20 0.40
GSK3A P49840 1/20 0.40
LIMK1 P53667 1/20 0.40
IKBKE Q14164 1/20 0.40
MAPK14 Q16539 1/20 0.40
TAOK1 Q7L7X3 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
DYRK1B Q9Y463 1/20 0.40
HRH4 Q9H3N8 2/20 0.35
REN P00797 8/20 0.33
SPR P35270 1/20 0.33
LRRK2 Q5S007 1/20 0.32
IKBKB O14920 1/20 0.32
TSHR P16473 1/20 0.32
GLA P06280 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21796485 0.78 CHEK1 (0.40) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL18399147 0.75 AXL (0.38) LIMK1
SCHEMBL5407783 0.75 CHEK1 (0.49) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL21797005 0.73 CHEK1 (0.47) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL21796894 0.72 IKBKB (0.41) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL21796483 0.71 CHEK1 (0.40) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL25313919 0.71 GABRP (0.40) HRH4RENTSHRGLA
SCHEMBL21796880 0.70 MAPT (0.44) LRRK2TSHR
SCHEMBL4787452 0.69 CHEK1 (0.54) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL21796520 0.69 CHEK1 (0.54) CHEK1AURKADAPK3CSNK1A1GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3325449-A1 COMPOUNDS GlaxoSmithKline Intellectual Property Development Limited (GB) 2018-05-30 EP disclosed
WO-2017012576-A1 COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-01-26 WO disclosed